SCHEMBL8634801

SCHEMBL8634801

CS(=O)(=O)c1cccn1-c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.46
PTGS2 P35354 5/20 0.44
ALDH1A1 P00352 3/20 0.41
MEN1 O00255 1/20 0.41
MAPT P10636 1/20 0.41
KMT2A Q03164 1/20 0.41
MCL1 Q07820 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
NOTUM Q6P988 1/20 0.38
DDB1 Q16531 1/20 0.37
CRBN Q96SW2 1/20 0.37
COMT P21964 1/20 0.37
SCN3A Q9NY46 1/20 0.37
KDM4E B2RXH2 2/20 0.36
CYP1A2 P05177 1/20 0.36
HPGD P15428 1/20 0.36
BLM P54132 1/20 0.36
HSD17B10 Q99714 1/20 0.36
GAA P10253 1/20 0.35
DRD2 P14416 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3262644 0.84 ATM (0.46) ATMPTGS2ALDH1A1MEN1MAPT
SCHEMBL28143996 0.82 ATM (0.47) ATMALDH1A1MEN1MAPTKMT2A
SCHEMBL5312009 0.72 PTGS2 (0.76) PTGS2
SCHEMBL14030743 0.70 TSHR (0.46) PTGS2ALDH1A1MEN1MAPTKMT2A
SCHEMBL7186907 0.68 CYP3A4 (0.44) PTGS2ALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL3433959 0.67 NOTUM (0.49) ALDH1A1MEN1MAPTKMT2ASMN1; SMN2
SCHEMBL28129191 0.67 ATM (0.48) ATMPTGS2ALDH1A1MEN1MAPT
SCHEMBL1127502 0.67 ATM (0.48) ATMALDH1A1MEN1MAPTKMT2A
SCHEMBL8505536 0.66 PTGS2 (0.39) PTGS2SMN1; SMN2NOTUMDDB1CRBN
SCHEMBL11101049 0.66 PSIP1 (0.41) ATMALDH1A1MEN1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0946507-A1 SUBSTITUTED PYRROLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1999-10-06 EP disclosed
WO-1998025896-A1 SUBSTITUTED PYRROLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1998-06-18 WO disclosed