SCHEMBL3434799

SCHEMBL3434799

CCOC(=O)Oc1cc(-c2cccc(C#N)c2)n(-c2ccc(F)c(Cl)c2)n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RPA1 P27694 3/20 0.42
RXFP1 Q9HBX9 1/20 0.41
MCHR1 Q99705 4/20 0.39
AR P10275 1/20 0.38
FAAH O00519 1/20 0.38
MGLL Q99685 1/20 0.38
CNR2 P34972 1/20 0.38
ADORA2A P29274 1/20 0.37
SLC16A3 O15427 1/20 0.37
SLC16A1 P53985 1/20 0.37
MCTS1 Q9ULC4 1/20 0.37
BRD9 Q9H8M2 1/20 0.37
RXRA P19793 1/20 0.36
RXRB P28702 1/20 0.36
RXRG P48443 1/20 0.36
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
MAPK1 P28482 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3432814 0.93 ALDH1A1 (0.38) RPA1RXFP1MCHR1KDM4EMEN1
SCHEMBL3434352 0.90 RPA1 (0.39) RPA1RXFP1BRD9RXRARXRB
SCHEMBL3433402 0.90 CNR2 (0.38) RPA1MCHR1FAAHMGLLCNR2
SCHEMBL1110649 0.90 ALDH1A1 (0.44) RPA1FAAHCNR2ADORA2ASLC16A3
SCHEMBL3427610 0.89 RPA1 (0.45) RPA1RXFP1ARFAAHMGLL
SCHEMBL3436334 0.88 CNR2 (0.43) RPA1FAAHMGLLCNR2ADORA2A
SCHEMBL3430605 0.88 RXFP1 (0.43) RPA1RXFP1FAAHBRD9ALDH1A1
SCHEMBL3434465 0.87 ALDH1A1 (0.44) RPA1SLC16A3SLC16A1MCTS1RXRA
SCHEMBL3434918 0.86 ALDH1A1 (0.40) RPA1FAAHMGLLSLC16A3SLC16A1
SCHEMBL1765280 0.85 CHRNA7 (0.50) RPA1RXFP1FAAHMGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2254885-A1 (PYRAZOLYL CARBONYL)IMIDAZOLIDINONE DERIVATIVES FOR THE TREATMENT OF RETROVIRAL DISEASES AiCuris GmbH & Co. KG (DE) 2010-12-01 EP disclosed
WO-2009115213-A1 (PYRAZOLYL CARBONYL)IMIDAZOLIDINONE DERIVATIVES FOR THE TREATMENT OF RETROVIRAL DISEASES AICURIS GMBH & CO. KG (DE) 2009-09-24 WO disclosed