SCHEMBL3434465

SCHEMBL3434465

CCOC(=O)Oc1cc(-c2cccc(Cl)c2)n(-c2cccc(C#N)c2)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.44
KDM4E B2RXH2 3/20 0.44
HTT P42858 2/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
MAPT P10636 1/20 0.44
MAPK1 P28482 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
TP53 P04637 2/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
RXRA P19793 3/20 0.41
RXRB P28702 3/20 0.41
RXRG P48443 3/20 0.41
DYRK3 O43781 1/20 0.41
DYRK1A Q13627 1/20 0.41
DYRK2 Q92630 1/20 0.41
DYRK1B Q9Y463 1/20 0.41
SLC16A3 O15427 1/20 0.41
SLC16A1 P53985 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1110649 0.97 ALDH1A1 (0.44) ALDH1A1KDM4EHTTMEN1KMT2A
SCHEMBL3436334 0.93 CNR2 (0.43) ALDH1A1KDM4ENPSR1TP53RPA1
SCHEMBL3434336 0.90 RXRA (0.40) ALDH1A1KDM4EHTTMEN1KMT2A
SCHEMBL3432814 0.89 ALDH1A1 (0.38) ALDH1A1KDM4EHTTMEN1KMT2A
SCHEMBL3434918 0.87 ALDH1A1 (0.40) ALDH1A1KDM4EHTTMEN1KMT2A
SCHEMBL3434799 0.87 RPA1 (0.42) ALDH1A1KDM4EHTTMEN1KMT2A
SCHEMBL3433370 0.87 ALDH1A1 (0.41) ALDH1A1KDM4EHTTMEN1KMT2A
SCHEMBL1110698 0.87 PPP1CA (0.50) ALDH1A1KDM4EHTTKMT2ATP53
SCHEMBL3430227 0.86 ALDH1A1 (0.45) ALDH1A1HTTTP53RXRARXRB
SCHEMBL3429282 0.86 FAAH (0.49) ALDH1A1KMT2ATP53SMN1; SMN2RXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2254885-A1 (PYRAZOLYL CARBONYL)IMIDAZOLIDINONE DERIVATIVES FOR THE TREATMENT OF RETROVIRAL DISEASES AiCuris GmbH & Co. KG (DE) 2010-12-01 EP disclosed
WO-2009115213-A1 (PYRAZOLYL CARBONYL)IMIDAZOLIDINONE DERIVATIVES FOR THE TREATMENT OF RETROVIRAL DISEASES AICURIS GMBH & CO. KG (DE) 2009-09-24 WO disclosed