SCHEMBL3433402

SCHEMBL3433402

CCOC(=O)Oc1cc(-c2cccc(C#N)c2)n(-c2ccc(F)c(C#N)c2)n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 1/20 0.38
MCHR1 Q99705 1/20 0.38
ADORA2A P29274 2/20 0.38
HRH2 P25021 1/20 0.36
HRH1 P35367 1/20 0.36
TLR8 Q9NR97 1/20 0.36
TLR7 Q9NYK1 1/20 0.36
PDE4D Q08499 1/20 0.36
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 2/20 0.35
HPGD P15428 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35
GABRA5 P31644 1/20 0.35
GABRA3 P34903 1/20 0.35
CYP1A2 P05177 1/20 0.35
GRM5 P41594 1/20 0.35
FNTA P49354 1/20 0.35
FNTB P49356 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3434918 0.92 ALDH1A1 (0.40) KDM4EALDH1A1SMN1; SMN2FAAHMGLL
SCHEMBL3434328 0.90 PGR (0.38) KDM4EALDH1A1HPGDSMN1; SMN2GRM5
SCHEMBL3434799 0.90 RPA1 (0.42) CNR2MCHR1ADORA2AHRH2HRH1
SCHEMBL3436334 0.89 CNR2 (0.43) CNR2ADORA2AHRH2HRH1TLR8
SCHEMBL1110649 0.87 ALDH1A1 (0.44) CNR2ADORA2AKDM4EALDH1A1HPGD
SCHEMBL1765512 0.85 CA9 (0.50) TLR8TLR7KDM4EALDH1A1HPGD
SCHEMBL3435607 0.85 RXRA (0.38) KDM4EALDH1A1FAAH
SCHEMBL3432814 0.85 ALDH1A1 (0.38) MCHR1KDM4EALDH1A1SMN1; SMN2RPA1
SCHEMBL3434266 0.84 PGR (0.39) CNR2ADORA2AHRH2HRH1TLR8
SCHEMBL3434465 0.84 ALDH1A1 (0.44) KDM4EALDH1A1HPGDSMN1; SMN2RPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2254885-A1 (PYRAZOLYL CARBONYL)IMIDAZOLIDINONE DERIVATIVES FOR THE TREATMENT OF RETROVIRAL DISEASES AiCuris GmbH & Co. KG (DE) 2010-12-01 EP disclosed
WO-2009115213-A1 (PYRAZOLYL CARBONYL)IMIDAZOLIDINONE DERIVATIVES FOR THE TREATMENT OF RETROVIRAL DISEASES AICURIS GMBH & CO. KG (DE) 2009-09-24 WO disclosed