SCHEMBL3436334

SCHEMBL3436334

CCOC(=O)Oc1cc(-c2cccc(C#N)c2)n(-c2cccc(C#N)c2)n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 1/20 0.43
ADORA2A P29274 2/20 0.42
HRH2 P25021 1/20 0.41
HRH1 P35367 1/20 0.41
ALDH1A1 P00352 3/20 0.41
KDM4E B2RXH2 2/20 0.41
HPGD P15428 1/20 0.41
GABRG2 P18507 1/20 0.40
GABRB3 P28472 1/20 0.40
GABRA5 P31644 1/20 0.40
GABRA3 P34903 1/20 0.40
TLR8 Q9NR97 1/20 0.40
TLR7 Q9NYK1 1/20 0.40
PDCD1 Q15116 1/20 0.39
CD274 Q9NZQ7 1/20 0.39
F11 P03951 1/20 0.39
FNTA P49354 1/20 0.39
FNTB P49356 1/20 0.39
TP53 P04637 1/20 0.39
TSHR P16473 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1110649 0.94 ALDH1A1 (0.44) CNR2ADORA2AALDH1A1KDM4EHPGD
SCHEMBL3434465 0.93 ALDH1A1 (0.44) ALDH1A1KDM4EHPGDTP53NPSR1
SCHEMBL3434266 0.91 PGR (0.39) CNR2ADORA2AHRH2HRH1ALDH1A1
SCHEMBL3433402 0.89 CNR2 (0.38) CNR2ADORA2AHRH2HRH1ALDH1A1
SCHEMBL3434799 0.88 RPA1 (0.42) CNR2ADORA2AHRH2HRH1ALDH1A1
SCHEMBL3432814 0.88 ALDH1A1 (0.38) ALDH1A1KDM4ETP53NPSR1RPA1
SCHEMBL3434336 0.87 RXRA (0.40) CNR2ALDH1A1KDM4EHPGDPDCD1
SCHEMBL3433370 0.84 ALDH1A1 (0.41) ALDH1A1KDM4ETP53NPSR1
SCHEMBL1765264 0.83 CA9 (0.54) ALDH1A1KDM4EHPGDTLR8TLR7
SCHEMBL1110698 0.81 PPP1CA (0.50) ALDH1A1KDM4ETP53FAAHRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2254885-A1 (PYRAZOLYL CARBONYL)IMIDAZOLIDINONE DERIVATIVES FOR THE TREATMENT OF RETROVIRAL DISEASES AiCuris GmbH & Co. KG (DE) 2010-12-01 EP disclosed
WO-2009115213-A1 (PYRAZOLYL CARBONYL)IMIDAZOLIDINONE DERIVATIVES FOR THE TREATMENT OF RETROVIRAL DISEASES AICURIS GMBH & CO. KG (DE) 2009-09-24 WO disclosed