SCHEMBL3440893

SCHEMBL3440893

COc1cccc(-c2nc3ccc(C4=NNC(=O)SC4C)cc3[nH]2)c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FBP1 P09467 1/20 0.59
ABCB11 O95342 1/20 0.56
MAOA P21397 1/20 0.56
ADORA2A P29274 1/20 0.56
PDE3B Q13370 1/20 0.56
PDE3A Q14432 1/20 0.56
NPC1 O15118 4/20 0.49
RAB9A P51151 3/20 0.49
TP53 P04637 3/20 0.49
HPGD P15428 3/20 0.49
POLB P06746 3/20 0.49
MEN1 O00255 2/20 0.49
PKM P14618 2/20 0.49
KMT2A Q03164 2/20 0.49
HTT P42858 1/20 0.49
ALDH1A1 P00352 3/20 0.48
SMN1; SMN2 Q16637 3/20 0.48
KDM4E B2RXH2 2/20 0.48
TSHR P16473 1/20 0.48
NFKB1 P19838 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3440912 0.92 FBP1 (0.50) FBP1ABCB11MAOAADORA2APDE3B
SCHEMBL3440988 0.82 FBP1 (0.56) FBP1ABCB11MAOAADORA2APDE3B
SCHEMBL3440867 0.82 FBP1 (0.56) FBP1ABCB11MAOAADORA2APDE3B
SCHEMBL3440983 0.80 FBP1 (0.66) FBP1ABCB11MAOAADORA2APDE3B
SCHEMBL3603104 0.79 GPR119 (0.42) FBP1PDE3BPDE3ANPC1RAB9A
SCHEMBL3440936 0.74 FBP1 (0.48) FBP1ABCB11MAOAADORA2APDE3B
SCHEMBL3440914 0.74 FBP1 (0.48) FBP1ABCB11MAOAADORA2APDE3B
SCHEMBL3609382 0.74 FBP1 (0.48) FBP1ABCB11MAOAADORA2APDE3B
Hydrochloric Acid SCHEMBL3618780 0.74 FBP1 (0.47) FBP1ABCB11MAOAADORA2APDE3B
Hydrochloric Acid SCHEMBL3440981 0.74 FBP1 (0.47) FBP1ABCB11MAOAADORA2APDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2229385-A2 BENZIMIDAZOLEDIHYDROTHIADIAZINONE DERIVATIVES AS FRUCTOSE-1,6-BISPHOSPHATASE INHIBITORS, AND PHARMACEUTICAL COMPOSITIONS COMPRISING SAME Merck Patent GmbH (DE) 2010-09-22 EP claimed
WO-2009062576-A2 BENZIMIDAZOLEDIHYDROTHIADIAZINONE DERIVATIVES AS FRUCTOSE-1,6-BISPHOSPHATASE INHIBITORS, AND PHARMACEUTICAL COMPOSITIONS COMPRISING SAME MERCK PATENT GMBH (DE) 2009-05-22 WO claimed
EP-2229385-A2 BENZIMIDAZOLEDIHYDROTHIADIAZINONE DERIVATIVES AS FRUCTOSE-1,6-BISPHOSPHATASE INHIBITORS, AND PHARMACEUTICAL COMPOSITIONS COMPRISING SAME Merck Patent GmbH (DE) 2010-09-22 EP disclosed
WO-2009062576-A2 BENZIMIDAZOLEDIHYDROTHIADIAZINONE DERIVATIVES AS FRUCTOSE-1,6-BISPHOSPHATASE INHIBITORS, AND PHARMACEUTICAL COMPOSITIONS COMPRISING SAME MERCK PATENT GMBH (DE) 2009-05-22 WO disclosed