SCHEMBL3440983

SCHEMBL3440983

CC1SC(=O)NN=C1c1ccc2nc(-c3ccc(N(C)C)cc3)[nH]c2c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FBP1 P09467 1/20 0.66
TCF4 P15884 1/20 0.53
CTNNB1 P35222 1/20 0.53
PDE3B Q13370 7/20 0.49
PDE3A Q14432 7/20 0.49
ABCB11 O95342 1/20 0.49
MAOA P21397 1/20 0.49
ADORA2A P29274 1/20 0.49
SIRT2 Q8IXJ6 1/20 0.47
SIRT1 Q96EB6 1/20 0.47
AURKA O14965 2/20 0.46
PDE4A P27815 5/20 0.45
PDE4B Q07343 5/20 0.45
PDE4C Q08493 5/20 0.45
PDE4D Q08499 5/20 0.45
F10 P00742 1/20 0.45
KDM4E B2RXH2 1/20 0.42
NPC1 O15118 1/20 0.42
GUSB P08236 1/20 0.42
MAPT P10636 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3613333 0.92 FBP1 (0.55) FBP1TCF4CTNNB1PDE3BPDE3A
SCHEMBL3440893 0.80 FBP1 (0.59) FBP1PDE3BPDE3AABCB11MAOA
SCHEMBL3440919 0.78 FBP1 (0.62) FBP1PDE3BPDE3AABCB11MAOA
SCHEMBL3440867 0.77 FBP1 (0.56) FBP1PDE3BPDE3AABCB11MAOA
SCHEMBL3440988 0.77 FBP1 (0.56) FBP1PDE3BPDE3AABCB11MAOA
SCHEMBL8767834 0.77 TCF4 (0.78) TCF4CTNNB1SIRT2SIRT1AURKA
SCHEMBL3441010 0.77 FBP1 (0.55) FBP1PDE3BPDE3AABCB11MAOA
SCHEMBL3614084 0.76 FBP1 (0.55) FBP1PDE3BPDE3AABCB11MAOA
SCHEMBL9182933 0.74 FBP1 (0.53) FBP1PDE3BPDE3APDE4APDE4B
SCHEMBL3602033 0.73 FBP1 (0.59) FBP1PDE3BPDE3AABCB11MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2229385-A2 BENZIMIDAZOLEDIHYDROTHIADIAZINONE DERIVATIVES AS FRUCTOSE-1,6-BISPHOSPHATASE INHIBITORS, AND PHARMACEUTICAL COMPOSITIONS COMPRISING SAME Merck Patent GmbH (DE) 2010-09-22 EP claimed
WO-2009062576-A2 BENZIMIDAZOLEDIHYDROTHIADIAZINONE DERIVATIVES AS FRUCTOSE-1,6-BISPHOSPHATASE INHIBITORS, AND PHARMACEUTICAL COMPOSITIONS COMPRISING SAME MERCK PATENT GMBH (DE) 2009-05-22 WO claimed