SCHEMBL3454176

SCHEMBL3454176

CC(C)CNC(=O)c1ccc2ccc(C(N)=O)cc2c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.59
GAA P10253 1/20 0.59
HSD17B10 Q99714 1/20 0.59
HPGD P15428 3/20 0.57
KDM4E B2RXH2 2/20 0.57
F3 P13726 4/20 0.50
MLYCD O95822 1/20 0.50
NPSR1 Q6W5P4 1/20 0.49
PRSS1 P07477 2/20 0.47
PRSS2 P07478 2/20 0.47
PRSS3 P35030 2/20 0.47
LCK P06239 1/20 0.47
PLAU P00749 3/20 0.47
OPRM1 P35372 1/20 0.44
OPRD1 P41143 1/20 0.44
RAB9A P51151 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
MEN1 O00255 1/20 0.43
MAPK14 Q16539 1/20 0.43
F2 P00734 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3033837 0.86 KMT2A (0.61) KMT2AGAAHSD17B10HPGDKDM4E
SCHEMBL16866256 0.84 GAA (0.68) KMT2AGAAHSD17B10HPGDKDM4E
SCHEMBL3028838 0.81 KMT2A (0.63) KMT2AGAAHSD17B10HPGDKDM4E
SCHEMBL3453839 0.78 HPGD (0.55) KMT2AHPGDKDM4EPRSS1LCK
SCHEMBL17865783 0.78 MLYCD (0.73) KMT2AGAAHSD17B10HPGDKDM4E
SCHEMBL6273049 0.77 GAA (0.66) KMT2AGAAHSD17B10HPGDKDM4E
SCHEMBL5482854 0.77 GAA (0.61) KMT2AGAAHSD17B10HPGDKDM4E
SCHEMBL10324044 0.77 HPGD (0.71) KMT2AGAAHSD17B10HPGDKDM4E
SCHEMBL3946696 0.76 KDM4E (0.75) KMT2AGAAHSD17B10HPGDKDM4E
SCHEMBL30935786 0.76 LCK (0.75) KMT2AHSD17B10KDM4EPRSS1LCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2205070-A1 N-HYDROXY-NAPHTHALENE DICARBOXAMIDE AND N-HYDROXY-BIPHENYL-DICARBOXAMIDE COMPOUNDS AS HISTONE DEACETYLASE INHIBITORS Merck Sharp & Dohme Corp. (US) 2010-07-14 EP claimed
WO-2009045385-A1 N-HYDROXY-NAPHTHALENE DICARBOXAMIDE AND N-HYDROXY-BIPHENYL-DICARBOXAMIDE COMPOUNDS AS HISTONE DEACETYLASE INHIBITORS MERCK & CO., INC. (US) 2009-04-09 WO claimed