SCHEMBL3454346

SCHEMBL3454346

Cc1nc(C#Cc2ccc(O)cc2)sc1C(=O)NC(C)c1ccc(F)cc1

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.50
PDE2A O00408 1/20 0.43
PTGER4 P35408 1/20 0.42
GABRA5 P31644 2/20 0.41
MAOA P21397 1/20 0.41
ACACB O00763 5/20 0.40
NPC1 O15118 1/20 0.40
KMT2A Q03164 1/20 0.40
LMNA P02545 1/20 0.40
STAT3 P40763 1/20 0.39
TSHR P16473 1/20 0.38
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13541870 0.89 ALDH1A1 (0.49) ALDH1A1ACACBLMNATSHRHTT
SCHEMBL3455839 0.87 HTT (0.46) ALDH1A1PDE2APTGER4ACACBNPC1
SCHEMBL3454459 0.80 SCD (0.55) LMNAHTT
SCHEMBL3447237 0.78 SCD (0.56) ALDH1A1NPC1LMNA
SCHEMBL13541863 0.77 ALDH1A1 (0.58) ALDH1A1PDE2AGABRA5MAOANPC1
SCHEMBL3454764 0.76 SCD (0.44) ALDH1A1NPC1KMT2ALMNA
SCHEMBL3455193 0.72 ATM (0.46) NPC1KMT2AHTT
SCHEMBL13494840 0.71 NPC1 (0.74) ALDH1A1MAOANPC1KMT2ALMNA
SCHEMBL3454348 0.70 SCD (0.55)
SCHEMBL16190459 0.70 ACACB (0.55) ALDH1A1ACACBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010007482-A2 THIAZOLE DERIVATIVES AS STEAROYL COA DESATURASE INHIBITORS GLENMARK PHARMACEUTICALS S.A. (CH) 2010-01-21 WO claimed
WO-2010007482-A2 THIAZOLE DERIVATIVES AS STEAROYL COA DESATURASE INHIBITORS GLENMARK PHARMACEUTICALS S.A. (CH) 2010-01-21 WO disclosed
WO-2010007482-A2 THIAZOLE DERIVATIVES AS STEAROYL COA DESATURASE INHIBITORS GLENMARK PHARMACEUTICALS S.A. (CH) 2010-01-21 WO disclosed