SCHEMBL3454483

SCHEMBL3454483

COc1ccc(NC(=O)c2ccc3ccc(C(N)=O)cc3c2)cc1

nearest known ligand 0.77

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 7/20 0.77
RAB9A P51151 7/20 0.77
CASP3 P42574 2/20 0.77
SENP7 Q9BQF6 2/20 0.77
PLAU P00749 12/20 0.75
PLAT P00750 4/20 0.72
PLG P00747 4/20 0.70
SMN1; SMN2 Q16637 4/20 0.65
TP53 P04637 3/20 0.65
ALOX15 P16050 1/20 0.65
F2 P00734 1/20 0.62
KLKB1 P03952 1/20 0.62
PRSS1 P07477 1/20 0.62
ALDH1A1 P00352 1/20 0.58
MAPT P10636 1/20 0.56
NQO2 P16083 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3036351 0.87 NPC1 (0.79) NPC1RAB9ACASP3SENP7PLAU
SCHEMBL3788361 0.87 NPC1 (1.00) NPC1RAB9ACASP3SENP7PLAU
SCHEMBL15412987 0.86 NPC1 (0.68) NPC1RAB9ACASP3SENP7PLAU
SCHEMBL15580882 0.84 NPC1 (0.74) NPC1RAB9ACASP3SENP7PLAU
SCHEMBL15031541 0.83 NPC1 (0.76) NPC1RAB9ACASP3SENP7PLAU
SCHEMBL28013893 0.81 PLAU (0.74) PLAUPLATPLGF2KLKB1
SCHEMBL21446854 0.81 PLAU (0.79) NPC1RAB9ACASP3SENP7PLAU
SCHEMBL5016280 0.81 PLAU (0.75) NPC1RAB9ACASP3SENP7PLAU
SCHEMBL6799157 0.80 RAB9A (1.00) NPC1RAB9ACASP3SENP7PLAU
SCHEMBL2917029 0.78 NPC1 (0.82) NPC1RAB9ACASP3SENP7PLAU

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2205070-A1 N-HYDROXY-NAPHTHALENE DICARBOXAMIDE AND N-HYDROXY-BIPHENYL-DICARBOXAMIDE COMPOUNDS AS HISTONE DEACETYLASE INHIBITORS Merck Sharp & Dohme Corp. (US) 2010-07-14 EP claimed
WO-2009045385-A1 N-HYDROXY-NAPHTHALENE DICARBOXAMIDE AND N-HYDROXY-BIPHENYL-DICARBOXAMIDE COMPOUNDS AS HISTONE DEACETYLASE INHIBITORS MERCK & CO., INC. (US) 2009-04-09 WO claimed