SCHEMBL3454742

SCHEMBL3454742

Cc1cc(Cc2c(C(N)=O)ccc3cc(C(N)=O)ccc23)no1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MBOAT4 Q96T53 1/20 0.37
LCK P06239 1/20 0.35
ADORA2A P29274 1/20 0.34
ADORA1 P30542 1/20 0.34
METAP2 P50579 1/20 0.34
KCNH2 Q12809 1/20 0.34
GRM2 Q14416 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
USP2 O75604 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
ALOX15 P16050 1/20 0.33
HSD17B10 Q99714 1/20 0.33
POLB P06746 1/20 0.33
EPHX2 P34913 1/20 0.33
AR P10275 1/20 0.33
KMT2A Q03164 1/20 0.33
PLAU P00749 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3454745 0.75 ROCK2 (0.52) ADORA2AADORA1NPC1RAB9AMAPT
SCHEMBL28217927 0.74 PLA2G4A (0.41) LCKNPC1ALDH1A1MAPTPOLB
SCHEMBL3031953 0.71 LCK (0.39) LCKMETAP2SMN1; SMN2NPC1RAB9A
SCHEMBL1568383 0.71 MBOAT4 (0.52) MBOAT4SMN1; SMN2NPC1RAB9AALDH1A1
SCHEMBL3028424 0.71 LCK (0.49) LCKSMN1; SMN2ALDH1A1MAPTHSD17B10
SCHEMBL15389131 0.70 NPC1 (0.43) SMN1; SMN2NPC1RAB9AUSP2ALDH1A1
SCHEMBL3454125 0.68 PLAU (0.43) PLAU
SCHEMBL29625781 0.67 LCK (0.56) LCKALDH1A1MAPTHSD17B10POLB
SCHEMBL1767492 0.67 SIRT3 (0.44) METAP2NPC1RAB9AUSP2ALDH1A1
SCHEMBL3454173 0.66 LCK (0.55) LCKALDH1A1MAPTPLAUKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2205070-A1 N-HYDROXY-NAPHTHALENE DICARBOXAMIDE AND N-HYDROXY-BIPHENYL-DICARBOXAMIDE COMPOUNDS AS HISTONE DEACETYLASE INHIBITORS Merck Sharp & Dohme Corp. (US) 2010-07-14 EP claimed
WO-2009045385-A1 N-HYDROXY-NAPHTHALENE DICARBOXAMIDE AND N-HYDROXY-BIPHENYL-DICARBOXAMIDE COMPOUNDS AS HISTONE DEACETYLASE INHIBITORS MERCK & CO., INC. (US) 2009-04-09 WO claimed