SCHEMBL3457587

SCHEMBL3457587

Cc1cnc(Cn2c(=O)[nH]c3sccc3c2=O)cn1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERCC1 P07992 1/20 0.45
ERCC5 P28715 1/20 0.45
FEN1 P39748 1/20 0.45
ERCC4 Q92889 1/20 0.45
ADRA1B P35368 2/20 0.42
ADRA1D P25100 1/20 0.42
ADRA1A P35348 1/20 0.42
TLR7 Q9NYK1 2/20 0.42
ALDH1A1 P00352 3/20 0.41
KDM4E B2RXH2 2/20 0.41
CDC7 O00311 1/20 0.36
MAPK13 O15264 1/20 0.36
DAPK3 O43293 1/20 0.36
ROCK2 O75116 1/20 0.36
MAP4K4 O95819 1/20 0.36
PIM1 P11309 1/20 0.36
GSK3A P49840 1/20 0.36
GSK3B P49841 1/20 0.36
NEK4 P51957 1/20 0.36
MAPK12 P53778 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2772730 0.79 QPCT (0.47) TLR7ALDH1A1KDM4EPARGHPGD
SCHEMBL24570158 0.78 PARG (0.49) ERCC1ERCC5FEN1ERCC4ADRA1B
SCHEMBL24570832 0.76 PARG (0.48) ERCC1ERCC5FEN1ERCC4ADRA1B
SCHEMBL2759479 0.74 ERCC1 (0.58) ERCC1ERCC5FEN1ERCC4ADRA1B
SCHEMBL6510464 0.73 ALDH1A1 (0.59) ERCC1ERCC5FEN1ERCC4ADRA1B
SCHEMBL26606602 0.73 ERCC1 (0.45) ERCC1ERCC5FEN1ERCC4ADRA1B
SCHEMBL10272797 0.69 ERCC1 (0.49) ERCC1ERCC5FEN1ERCC4ADRA1B
SCHEMBL24570735 0.68 ADRA1B (0.42) ERCC1ERCC5FEN1ERCC4ADRA1B
SCHEMBL6518727 0.68 FEN1 (0.47) ERCC1ERCC5FEN1ERCC4ADRA1B
SCHEMBL2733484 0.68 ERCC1 (0.50) ERCC1ERCC5FEN1ERCC4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2253630-A1 Heterocyclic compound and use thereof Takeda Pharmaceutical Company Limited (JP) 2010-11-24 EP disclosed