Mazaticol

Mazaticol

SCHEMBL34619

CN1[C@@H]2CCC(C)(C)[C@H]1C[C@H](OC(=O)C(O)(c1cccs1)c1cccs1)C2

nearest known ligand 0.51

Full drug profile on Sugi Atlas →

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 19/20 0.51
CHRM2 P08172 14/20 0.51
CHRM1 P11229 12/20 0.49
CHRM4 P08173 3/20 0.49
CHRM5 P08912 3/20 0.49
TSPO P30536 1/20 0.49
ADRA1A P35348 1/20 0.49
HRH1 P35367 1/20 0.49
OPRK1 P41145 1/20 0.49
KCNH2 Q12809 1/20 0.49
PDE3A Q14432 1/20 0.49
TMEM97 Q5BJF2 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Mazaticol SCHEMBL182361 0.99 CHRM3 (0.50) CHRM3CHRM2CHRM1CHRM4CHRM5
Mazaticol SCHEMBL17747972 0.98 CHRM3 (0.50) CHRM3CHRM2CHRM1CHRM4CHRM5
SCHEMBL4886970 0.86 CHRM3 (0.60) CHRM3CHRM2CHRM1CHRM4CHRM5
SCHEMBL4886984 0.86 CHRM3 (0.60) CHRM3CHRM2CHRM1CHRM4CHRM5
SCHEMBL4886957 0.86 CHRM3 (0.60) CHRM3CHRM2CHRM1CHRM4CHRM5
Mazaticol SCHEMBL15229491 0.84 ADRA1A (0.39) CHRM3CHRM2CHRM1CHRM4CHRM5
Mazaticol SCHEMBL28086106 0.79 CHRM3 (0.34) CHRM3CHRM2CHRM1CHRM4CHRM5
SCHEMBL16742011 0.77 CHRM3 (0.60) CHRM3CHRM2CHRM1CHRM4CHRM5
SCHEMBL14472825 0.77 CHRM3 (0.60) CHRM3CHRM2CHRM1CHRM4CHRM5
SCHEMBL1900207 0.77 CHRM3 (0.60) CHRM3CHRM2CHRM1CHRM4CHRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 480 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4154879-B1 PHARMACEUTICAL COMPOSITION FOR PREVENTING OR TREATING NICOTINE WITHDRAWAL SYMPTOMS KOREA INST SCI & TECH (KR) 2025-09-10 EP claimed
US-12350261-B2 Methods and devices for the treatment of ocular diseases in human subjects CLEARSIDE BIOMEDICAL, INC. (US) 2025-07-08 US claimed
WO-2025038382-A1 PHARMACEUTICAL ADHESIVE COMPOSITIONS MOMENTIVE PERFORMANCE MATERIALS INC. (US) 2025-02-20 WO claimed
WO-2024218296-A1 COMBINATION TREATMENTS COMPRISING ADMINISTRATION OF LEUCINE-RICH REPEAT KINASE 2 (LRRK2) INHIBITORS H. LUNDBECK A/S (DK) 2024-10-24 WO claimed
US-12102653-B2 Ligand regulated protein-protein interaction system ST. ANNA KINDERKREBSFORSCHUNG (AT) 2024-10-01 US claimed
US-20240000841-A1 LIGAND REGULATED PROTEIN-PROTEIN INTERACTION SYSTEM ST ANNA KINDERKREBSFORSCHUNG (AT) 2024-01-04 US claimed
US-11844813-B2 Ligand regulated protein-protein interaction system ST. ANNA KINDERKREBSFORSCHUNG (AT) 2023-12-19 US claimed
EP-4154879-A1 PHARMACEUTICAL COMPOSITION FOR PREVENTING OR TREATING NICOTINE WITHDRAWAL SYMPTOMS Korea Institute of Science and Technology (KR) 2023-03-29 EP claimed
EP-3852608-A1 COMPOSITIONS AND METHODS FOR GLAUCOMA Aufbau Medical Innovations Limited (IE) 2021-07-28 EP claimed
US-10987316-B2 Compositions and methods for transdermal delivery of tertiary amine drugs NOVEN PHARMACEUTICALS, INC. (US) 2021-04-27 US claimed
EP-2586401-A1 Implantable film/mesh composite Covidien LP (US) 2013-05-01 EP claimed
EP-2586607-A1 Implantable film/mesh composite for passage of tissue therebetween Covidien LP (US) 2013-05-01 EP claimed
US-20130102959-A1 Implantable Film/Mesh Composite COVIDIEN LP (US) 2013-04-25 US claimed
US-20130103060-A1 Implantable Film/Mesh Composite COVIDIEN LP (US) 2013-04-25 US claimed
US-20130030360-A1 Implantable Devices Including A Mesh And A Pivotable Film TYCO HEALTHCARE GROUP LP, (US) 2013-01-31 US claimed
US-20100226943-A1 SURFACE TOPOGRAPHIES FOR NON-TOXIC BIOADHESION CONTROL UNIVERSITY OF FLORIDA (US) 2010-09-09 US claimed
CN-101330905-A Freeze-drying process and products obtained thereby SCIDOSE LLC (US) 2008-12-24 CN claimed
EP-1954244-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY Scidose, Llc (US) 2008-08-13 EP claimed
WO-2007061529-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY SCIDOSE LLC. (US) 2007-05-31 WO claimed
US-20070116729-A1 Lyophilization process and products obtained thereby SCIDOSE LLC 2007-05-24 US claimed