Benzene

Benzene

SCHEMBL3466087

Nc1cccnn1.c1ccccc1

nearest known ligand 0.46

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GOT1 P17174 1/20 0.46
NOS3 P29474 3/20 0.42
NOS2 P35228 3/20 0.42
NOS1 P29475 2/20 0.42
PI4KA P42356 1/20 0.42
PI4K2B Q8TCG2 1/20 0.42
PI4K2A Q9BTU6 1/20 0.42
PI4KB Q9UBF8 1/20 0.42
P2RX7 Q99572 1/20 0.39
CYP1A2 P05177 1/20 0.38
BCAT2 O15382 1/20 0.35
ASIC3 Q9UHC3 1/20 0.34
NAPRT Q6XQN6 1/20 0.32
KDM4E B2RXH2 2/20 0.32
TSHR P16473 1/20 0.32
HDAC4 P56524 1/20 0.31
HSP90AA1 P07900 1/20 0.30
GRM4 Q14833 1/20 0.30
ALDH1A1 P00352 1/20 0.30
EPHX2 P34913 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26878 0.97
SCHEMBL30068488 0.97
Hydrochloric Acid SCHEMBL30294929 0.94 GOT1 (0.46) GOT1NOS3NOS2NOS1PI4KA
Hydrochloric Acid SCHEMBL4709475 0.94 GOT1 (0.46) GOT1NOS3NOS2NOS1PI4KA
SCHEMBL30711694 0.94
Hydrochloric Acid SCHEMBL753209 0.94
Hydrochloric Acid SCHEMBL3974934 0.94
Hydrazine SCHEMBL11032075 0.94
Biphenyl SCHEMBL27923035 0.91 ASIC3 (0.43) GOT1NOS3NOS2NOS1PI4KA
Acetic Acid SCHEMBL28012854 0.87 P2RX7 (0.44) GOT1NOS3NOS2NOS1PI4KA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8791116-B2 Myosin light chain kinase inhibitor compounds, compositions and related methods of use NORTHWESTERN UNIVERSITY (US) 2014-07-29 US disclosed
US-20130029999-A1 MYOSIN LIGHT CHAIN KINASE INHIBITOR COMPOUNDS, COMPOSITIONS AND RELATED METHODS OF USE NORTHWESTERN UNIVERSITY (US) 2013-01-31 US disclosed
US-8278305-B2 Myosin light chain kinase inhibitor compounds, compositions and related methods of use NORTHWESTERN UNIVERSITY (US) 2012-10-02 US disclosed
US-20100240668-A1 Myosin Light Chain Kinase Inhibitor Compounds, Compositions and Related Methods of Use NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2010-09-23 US disclosed
US-7732445-B2 Myosin light chain kinase inhibitor compounds, compostions and related methods of use NORTHWESTERN UNIVERSITY (US) 2010-06-08 US disclosed
WO-2008011176-A9 MYOSIN LIGHT CHAIN KINASE INHIBITOR COMPOUNDS, COMPOSITIONS AND RELATED METHODS OF USE UNIV NORTHWESTERN (US) 2008-03-06 WO disclosed
WO-2008011176-A2 MYOSIN LIGHT CHAIN KINASE INHIBITOR COMPOUNDS, COMPOSITIONS AND RELATED METHODS OF USE NORTHWESTERN UNIVERSITY (US) 2008-01-24 WO disclosed
US-20080021035-A1 Myosin light chain kinase inhibitor compounds, compostions and related methods of use NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2008-01-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130029999-A1 MYOSIN LIGHT CHAIN KINASE INHIBITOR COMPOUNDS, COMPOSITIONS AND RELATED METHODS OF USE MYLK, MYLK2, MYLK3 GOT1 3030/4885NOS3 3501/4885NOS2 3833/4885
US-20080021035-A1 Myosin light chain kinase inhibitor compounds, compostions and related methods of use MYLK, MYLK3, MYLK2 GOT1 3847/4885NOS3 2441/4885NOS2 2662/4885
US-20100240668-A1 Myosin Light Chain Kinase Inhibitor Compounds, Compositions and Related Methods of Use MYLK, MYLK2, MYLK3 GOT1 3030/4885NOS3 3501/4885NOS2 3833/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.