SCHEMBL3466639

SCHEMBL3466639

O=C1[C]Cc2cc(-c3ccc(Cl)c(C(F)(F)F)c3)ccc2N1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 9/20 0.45
CYP1A2 P05177 1/20 0.45
KIF11 P52732 1/20 0.45
PDE3B Q13370 2/20 0.43
PDE3A Q14432 2/20 0.43
PRF1 P14222 1/20 0.38
GRIA1 P42261 1/20 0.37
CACNG8 Q8WXS5 1/20 0.37
PGR P06401 1/20 0.36
AR P10275 1/20 0.36
ABL1 P00519 1/20 0.36
BCR P11274 1/20 0.36
COMT P21964 1/20 0.36
TDP2 O95551 1/20 0.36
KDR P35968 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3467162 0.82 KIF11 (0.65) NOTUMCYP1A2KIF11PDE3BPDE3A
SCHEMBL3312695 0.79 KIF11 (0.68) NOTUMCYP1A2KIF11PDE3BPDE3A
SCHEMBL3467329 0.75 KIF11 (0.46) NOTUMKIF11PDE3BPDE3AGRIA1
SCHEMBL3466905 0.72 OTUD7B (0.52) KIF11GRIA1CACNG8ABL1
SCHEMBL3467035 0.72 NOTUM (0.43) NOTUMCYP1A2PDE3BPDE3APRF1
SCHEMBL2698021 0.72 NOTUM (0.61) NOTUMCYP1A2PDE3BPDE3ACOMT
SCHEMBL4890959 0.68 KIF11 (0.68) CYP1A2KIF11PDE3BPDE3AGRIA1
SCHEMBL1899619 0.65 PDE3B (0.56) CYP1A2KIF11PDE3BPDE3AGRIA1
SCHEMBL700817 0.65 NOTUM (0.51) NOTUMCYP1A2PDE3BPDE3AAR
SCHEMBL18189320 0.64 KIF11 (0.58) CYP1A2KIF11PDE3BPDE3AGRIA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010074807-A1 3, 4-DIHYDROQUINOLIN-2 ( 1H ) -ONE DERIVATIVES AS SODIUM CHANNEL MODULATORS GILEAD PALO ALTO, INC. (US) 2010-07-01 WO disclosed