SCHEMBL3467035

SCHEMBL3467035

CC(C)(C)C1[C]C(=O)Nc2ccc(-c3ccc(Cl)c(C(F)(F)F)c3)cc21

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 10/20 0.43
CYP1A2 P05177 1/20 0.43
PDE3B Q13370 2/20 0.41
PDE3A Q14432 2/20 0.41
AR P10275 1/20 0.37
COMT P21964 1/20 0.37
PRF1 P14222 1/20 0.36
PGR P06401 2/20 0.36
KCNH2 Q12809 1/20 0.34
KDR P35968 1/20 0.34
SLC22A12 Q96S37 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3466639 0.72 NOTUM (0.45) NOTUMCYP1A2PDE3BPDE3AAR
SCHEMBL2698021 0.69 NOTUM (0.61) NOTUMCYP1A2PDE3BPDE3ACOMT
SCHEMBL3312695 0.66 KIF11 (0.68) NOTUMCYP1A2PDE3BPDE3APGR
SCHEMBL12508243 0.64 AR (0.57) NOTUMCYP1A2PDE3BPDE3AAR
SCHEMBL3034754 0.64 PDE3B (0.41) NOTUMCYP1A2PDE3BPDE3AAR
SCHEMBL700817 0.62 NOTUM (0.51) NOTUMCYP1A2PDE3BPDE3AAR
SCHEMBL1041571 0.62 NOTUM (0.53) NOTUMCYP1A2PDE3BPDE3AAR
SCHEMBL17297750 0.61 NOTUM (0.49) NOTUMCYP1A2PDE3BPDE3ACOMT
SCHEMBL693639 0.61 NOTUM (0.45) NOTUMCYP1A2PDE3BPDE3ACOMT
SCHEMBL19523185 0.61 CTSS (0.52) NOTUMKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010074807-A1 3, 4-DIHYDROQUINOLIN-2 ( 1H ) -ONE DERIVATIVES AS SODIUM CHANNEL MODULATORS GILEAD PALO ALTO, INC. (US) 2010-07-01 WO claimed