SCHEMBL3467567

SCHEMBL3467567

CC(C)(C)[Si](C)(C)OCCc1cc(C(N)=O)c(Br)cc1Cl

nearest known ligand 0.32

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.32
CA12 O43570 2/20 0.31
CA1 P00915 2/20 0.31
CA2 P00918 2/20 0.31
CA9 Q16790 2/20 0.31
CA14 Q9ULX7 2/20 0.31
CA3 P07451 1/20 0.31
CA4 P22748 1/20 0.31
CA6 P23280 1/20 0.31
CA5A P35218 1/20 0.31
CA7 P43166 1/20 0.31
CA13 Q8N1Q1 1/20 0.31
CA5B Q9Y2D0 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3468243 0.81 CA12 (0.31) CA12CA1CA2CA9CA14
SCHEMBL21356177 0.77 DUT (0.31) CA12CA1CA2CA9CA14
SCHEMBL3467792 0.74 CA12 (0.37) CA12CA1CA2CA9CA14
SCHEMBL13303932 0.74 ALDH1A1 (0.32)
SCHEMBL3344285 0.72 CA12 (0.40) KDM4ECA12CA1CA2CA9
SCHEMBL6114675 0.72 DUT (0.34) CA12CA1CA9
SCHEMBL3342503 0.72 APLNR (0.35) CA12CA1CA2CA9CA14
SCHEMBL3342251 0.71 TSHR (0.33) KDM4ECA12CA1CA2CA9
SCHEMBL21367294 0.70 DUT (0.37) CA12CA1CA2CA9CA14
SCHEMBL23883039 0.70 EPHX2 (0.39) CA12CA1CA2CA9CA14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2393781-A1 DIHYDROPYRIDONE UREAS AS P2X7 MODULATORS F. Hoffmann-La Roche AG (CH) 2011-12-14 EP disclosed
WO-2010072599-A1 DIHYDROPYRIDONE UREAS AS P2X7 MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2010-07-01 WO disclosed