SCHEMBL3467792

SCHEMBL3467792

NC(=O)c1cc(CCO)c(Cl)cc1Br

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 5/20 0.37
CA1 P00915 5/20 0.37
CA2 P00918 5/20 0.37
CA3 P07451 5/20 0.37
CA4 P22748 5/20 0.37
CA6 P23280 5/20 0.37
CA5A P35218 5/20 0.37
CA7 P43166 5/20 0.37
CA9 Q16790 5/20 0.37
CA13 Q8N1Q1 5/20 0.37
CA14 Q9ULX7 5/20 0.37
CA5B Q9Y2D0 5/20 0.37
KMT2A Q03164 2/20 0.35
ATM Q13315 1/20 0.35
SIRT1 Q96EB6 1/20 0.32
CASP1 P29466 1/20 0.32
DGAT1 O75907 1/20 0.32
MAPK8 P45983 1/20 0.31
NNMT P40261 1/20 0.31
ADRA1D P25100 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3344285 0.88 CA12 (0.40) CA12CA1CA2CA3CA4
SCHEMBL3342943 0.80 NNMT (0.37) CA12CA1CA2CA3CA4
SCHEMBL3342235 0.78 CA12 (0.46) CA12CA1CA2CA3CA4
SCHEMBL3468380 0.75 MEN1 (0.34) KMT2AMAPTALDH1A1NPSR1POLB
SCHEMBL3467567 0.74 KDM4E (0.32) CA12CA1CA2CA3CA4
SCHEMBL3342131 0.73 P2RX7 (0.37) CA12CA1CA2CA3CA4
SCHEMBL3339243 0.73 CA12 (0.46) CA12CA1CA2CA3CA4
SCHEMBL3339247 0.72 CA1 (0.41) CA12CA1CA2CA3CA4
SCHEMBL3339250 0.72 DGAT1 (0.47) CA12CA1CA2CA3CA4
SCHEMBL16644420 0.71 DGAT1 (0.46) CA12CA1CA2CA3CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2393781-A1 DIHYDROPYRIDONE UREAS AS P2X7 MODULATORS F. Hoffmann-La Roche AG (CH) 2011-12-14 EP disclosed
WO-2010072599-A1 DIHYDROPYRIDONE UREAS AS P2X7 MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2010-07-01 WO disclosed