SCHEMBL3477919

SCHEMBL3477919

COc1ccc2[nH]cc(C(N)=O)c(=O)c2c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.64
HSD17B10 Q99714 3/20 0.64
LMNA P02545 3/20 0.64
ALDH1A1 P00352 3/20 0.64
HPGD P15428 1/20 0.64
NR4A2 P43354 1/20 0.63
MEN1 O00255 2/20 0.60
KMT2A Q03164 2/20 0.60
MAPT P10636 2/20 0.60
MITF O75030 1/20 0.60
RAB9A P51151 1/20 0.60
NPSR1 Q6W5P4 1/20 0.60
CYP1A2 P05177 2/20 0.54
CYP2C19 P33261 2/20 0.54
CYP2C9 P11712 1/20 0.54
HTT P42858 1/20 0.54
MTNR1A P48039 1/20 0.53
MTNR1B P49286 1/20 0.53
HTR2B P41595 1/20 0.51
CPT1A P50416 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3633587 0.90 NR4A2 (0.73) KDM4EHSD17B10LMNAALDH1A1HPGD
SCHEMBL2053494 0.87 HTT (0.70) KDM4EHSD17B10LMNAALDH1A1HPGD
SCHEMBL29950498 0.86 LMNA (0.64) KDM4EHSD17B10LMNAALDH1A1HPGD
Hydrochloric Acid SCHEMBL7514852 0.86 HTT (0.68) KDM4EHSD17B10LMNAALDH1A1HPGD
SCHEMBL6204275 0.85 HTT (0.64) KDM4EHSD17B10LMNAALDH1A1HPGD
SCHEMBL28872023 0.83 KDM4E (0.61) KDM4EHSD17B10LMNAALDH1A1HPGD
SCHEMBL11101264 0.82 KDM4E (0.60) KDM4EHSD17B10LMNAALDH1A1HPGD
SCHEMBL9725707 0.82 LMNA (0.64) KDM4EHSD17B10LMNAALDH1A1HPGD
SCHEMBL3847939 0.81 GABRA1 (0.73) KDM4EHSD17B10LMNAALDH1A1HPGD
SCHEMBL28289149 0.81 SMN1; SMN2 (0.62) KDM4EHSD17B10LMNAALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010073078-A2 HETEROCYCLIC COMPOUNDS AS HDAC INHIBITORS ORCHID RESEARCH LABORATORIES LTD. (IN) 2010-07-01 WO claimed
EP-1177177-B1 SUBSTITUTED 4-OXO-QUINOLINE-3-CARBOXAMIDES: GABA BRAIN RECEPTOR LIGANDS NEUROGEN CORP (US) 2005-02-23 EP disclosed
US-6413956-B1 AGONISTS, ANTAGONISTS OR INVERSE AGONISTS AND LOCALIZATION PROBES FOR GAMMA AMINOBUTYRIC ACID BRAIN RECEPTORS; ANXIETY, DEPRESSION, DOWN SYNDROME, SLEEP AND SEIZURE DISORDERS, OVERDOSE WITH BENZODIAZEPINE DRUGS AND MEMORY ENHANCEMENT NEUROGEN CORPORATION 2002-07-02 US disclosed