SCHEMBL3478009

SCHEMBL3478009

COc1ccc(CN(c2ncns2)S(=O)(=O)c2cc(F)c(Oc3ccc(Cl)cc3-c3ccnn3C3CN(C(=O)O)C3C(C)(C)C)cc2F)c(OC)c1

nearest known ligand 0.49

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 20/20 0.49
CYP2C9 P11712 4/20 0.48
SCN5A Q14524 3/20 0.48
CYP3A4 P08684 2/20 0.48
SCN2B O60939 1/20 0.48
SCN1B Q07699 1/20 0.48
SCN1A P35498 1/20 0.37
SCN2A Q99250 1/20 0.37
SCN3A Q9NY46 1/20 0.37
SCN8A Q9UQD0 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1094239 0.87 SCN9A (0.52) SCN9ACYP2C9SCN5ACYP3A4SCN2B
SCHEMBL1094276 0.85 SCN9A (0.52) SCN9ACYP2C9SCN5ACYP3A4SCN2B
SCHEMBL9923647 0.81 SCN9A (0.51) SCN9ACYP2C9SCN5ACYP3A4SCN2B
SCHEMBL16011331 0.81 SCN9A (0.60) SCN9ACYP2C9SCN5ACYP3A4SCN2B
SCHEMBL9924685 0.80 SCN9A (0.44) SCN9ACYP2C9SCN5ACYP3A4SCN2B
SCHEMBL16011228 0.78 SCN9A (0.52) SCN9ACYP2C9SCN5ACYP3A4SCN1A
SCHEMBL1094117 0.77 SCN9A (0.53) SCN9ACYP2C9SCN5ACYP3A4SCN2B
SCHEMBL14933663 0.76 SCN9A (0.62) SCN9ACYP2C9SCN5A
SCHEMBL3477862 0.76 SCN9A (0.43) SCN9A
SCHEMBL14933655 0.76 SCN9A (0.59) SCN9ASCN1ASCN2ASCN3ASCN8A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100197655-A1 SULFONAMIDE DERIVATIVES Pfizer Limited Icagen, Inc. 2010-08-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100197655-A1 SULFONAMIDE DERIVATIVES SULT2A1, SULT1A1, TPST2 SCN9A 73/4885CYP2C9 75/4885SCN5A 19/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.