SCHEMBL3494044

SCHEMBL3494044

OS1(O)[CH]CCc2ccccc21

nearest known ligand 0.33

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.33
ORAI1 Q96D31 1/20 0.31
ORAI2 Q96SN7 1/20 0.31
ORAI3 Q9BRQ5 1/20 0.31
MAOA P21397 1/20 0.30
MAOB P27338 1/20 0.30
DRD2 P14416 1/20 0.30
DRD1 P21728 1/20 0.30
DRD4 P21917 1/20 0.30
DRD5 P21918 1/20 0.30
DRD3 P35462 1/20 0.30
HTR2C P28335 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL560871 0.77 ORAI1 (0.33) TSHRORAI1ORAI2ORAI3
SCHEMBL1463955 0.74 GPR3 (0.34) TSHRMAOAMAOBDRD2DRD1
SCHEMBL18065143 0.68 TSHR (0.42) TSHRORAI1ORAI2ORAI3MAOA
SCHEMBL3494049 0.65 TSHR (0.50) TSHRORAI1ORAI2ORAI3MAOA
SCHEMBL11777743 0.64 TSHR (0.41) TSHRORAI1ORAI2ORAI3MAOA
SCHEMBL7346113 0.63 CA12 (0.40) TSHR
SCHEMBL19820978 0.62 GPR3 (0.52) TSHRORAI1ORAI2ORAI3MAOA
SCHEMBL4166748 0.59 TSHR (0.56) TSHRORAI1ORAI2ORAI3MAOA
SCHEMBL862127 0.59 TSHR (0.56) TSHRORAI1ORAI2ORAI3MAOA
SCHEMBL862128 0.59 TSHR (0.56) TSHRORAI1ORAI2ORAI3MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100113418-A1 HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-05-06 US disclosed
EP-2123652-A1 HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2009-11-25 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100113418-A1 HETEROCYCLIC COMPOUND ACACA, ACAT1, CPT1B TSHR 3339/4885ORAI1 806/4885ORAI2 1923/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.