SCHEMBL350238

SCHEMBL350238

COc1ccc(C(CN)C[PH](=O)O)cc1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.47
L3MBTL1 Q9Y468 1/20 0.44
AOC3 Q16853 2/20 0.41
CYP2C19 P33261 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
SLC6A2 P23975 2/20 0.40
SLC6A4 P31645 2/20 0.40
SLC6A3 Q01959 1/20 0.40
FFAR1 O14842 1/20 0.39
CYP3A4 P08684 2/20 0.38
MEN1 O00255 1/20 0.38
MAPT P10636 1/20 0.38
PPARG P37231 1/20 0.38
KMT2A Q03164 1/20 0.38
ACP3 P15309 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL350645 0.81 GABBR2 (0.38) CYP2C19CYP1A2CYP2D6CYP3A4MEN1
SCHEMBL11079771 0.80 ALDH1A1 (0.54) ALDH1A1L3MBTL1AOC3CYP2C19CYP1A2
SCHEMBL349306 0.78 GABBR2 (0.56) CYP2C19CYP1A2CYP2D6CYP3A4MEN1
SCHEMBL351660 0.78 GABBR2 (0.57) CYP2C19CYP1A2CYP2D6SLC6A4SLC6A3
SCHEMBL350711 0.78 GABBR2 (0.56) CYP2C19CYP1A2CYP2D6SLC6A2SLC6A4
SCHEMBL5652935 0.75 ALDH1A1 (0.50) ALDH1A1L3MBTL1AOC3CYP2C19CYP1A2
SCHEMBL21465820 0.75 ALDH1A1 (0.50) ALDH1A1L3MBTL1AOC3CYP2C19CYP1A2
SCHEMBL10200947 0.75 GABBR2 (0.64) ALDH1A1L3MBTL1CYP2C19CYP1A2CYP2D6
SCHEMBL350431 0.74 CES2 (0.39) CYP2C19CYP1A2CYP2D6CYP3A4MEN1
SCHEMBL341858 0.73 ALDH1A1 (0.45) ALDH1A1L3MBTL1AOC3CYP2C19CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120016021-A1 METHODS OF TREATING FRAGILE X SYNDROME, DOWN'S SYNDROME, AUTISM AND RELATED DISORDERS XENOPORT, INC. (US) 2012-01-19 US disclosed
WO-2012009646-A1 METHODS OF TREATING FRAGILE X SYNDROME, DOWN'S SYNDROME, AUTISM AND RELATED DISORDERS XENOPORT, INC. (US) 2012-01-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120016021-A1 METHODS OF TREATING FRAGILE X SYNDROME, DOWN'S SYNDROME, AUTISM AND RELATED DISORDERS GABBR2, GABBR1, GABRB1 ALDH1A1 1156/4885L3MBTL1 2986/4885AOC3 2672/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.