SCHEMBL3525941

SCHEMBL3525941

CC(C)NS(=O)(=O)c1ccc(Cl)cc1C(=O)O

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.54
KDM4E B2RXH2 2/20 0.54
CHRM2 P08172 1/20 0.47
CHRM1 P11229 1/20 0.47
RRM1 P23921 1/20 0.47
RRM2B Q7LG56 1/20 0.47
ACLY P53396 1/20 0.47
ALDH1A1 P00352 1/20 0.46
TP53 P04637 1/20 0.46
HSD17B10 Q99714 1/20 0.45
GSTO1 P78417 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CNR2 P34972 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3521898 0.83 ALDH1A1 (0.50) KDM4EACLYALDH1A1TP53HSD17B10
SCHEMBL3525514 0.82 NPSR1 (0.54) NPSR1KDM4EALDH1A1GSTO1
SCHEMBL13543511 0.81 NPSR1 (0.52) NPSR1KDM4EACLYALDH1A1HSD17B10
SCHEMBL16000135 0.79 TRPV4 (0.51) ALDH1A1GSTO1CNR2
SCHEMBL26212920 0.78 CA1 (0.64) NPSR1KDM4EALDH1A1CA1CA2
SCHEMBL8489072 0.77 ALDH1A1 (0.55) KDM4EACLYALDH1A1TP53HSD17B10
SCHEMBL3523438 0.77 NPSR1 (0.61) NPSR1KDM4EHSD17B10GSTO1
SCHEMBL3526776 0.77 CA12 (0.65) ACLYALDH1A1
SCHEMBL16000114 0.76 MCL1 (0.57) KDM4EALDH1A1GSTO1
SCHEMBL3524715 0.75 ALDH1A1 (0.57) KDM4EACLYALDH1A1TP53HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7645771-B2 CCR5 antagonists as therapeutic agents SMITHKLINE BEECHAM CORP. (US) 2010-01-12 US disclosed
US-20060229336-A1 Ccr5 antagonists as therapeutic agents SMITHKLINE BEECHAM CORPORATION 2006-10-12 US disclosed
CN-1744899-A Piperidine derivatives as CCR5 antagonists SMITHKLINE BEECHAM CORP (US) 2006-03-08 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060229336-A1 Ccr5 antagonists as therapeutic agents CCR5, CCR1, CXCR3 NPSR1 338/4885KDM4E 4644/4885CHRM2 638/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.