SCHEMBL3528466

SCHEMBL3528466

CN=c1scc(CCl)n1C

nearest known ligand 0.42

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 1/20 0.39
ALDH1A1 P00352 2/20 0.36
GAA P10253 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6049077 1.00 CXCR4 (0.39) CXCR4ALDH1A1GAA
Hydrochloric Acid SCHEMBL3894282 0.98 CXCR4 (0.39) CXCR4ALDH1A1GAA
SCHEMBL3894363 0.70
Hydrochloric Acid SCHEMBL3909331 0.64 PDE4D (0.34) ALDH1A1
Hydrochloric Acid SCHEMBL3900671 0.62
Hydrochloric Acid SCHEMBL3901555 0.62 ALDH1A1 (0.40) ALDH1A1
Hydrochloric Acid SCHEMBL3901551 0.62 ALDH1A1 (0.40) ALDH1A1
Hydrochloric Acid SCHEMBL3908786 0.59
Hydrochloric Acid SCHEMBL3908782 0.59
Hydrochloric Acid SCHEMBL4823268 0.58 GPR84 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7671078-B2 Isothiourea derivatives of imadazo[2,1-b]Thiazoles and 5,6-dihydro derivatives thereof useful as CXCR4 chemokine receptor inhibitors NOVARTIS AG (CH) 2010-03-02 US disclosed
US-20070161618-A1 Isothiourea derivatives NOVARTIS AG (CH) 2007-07-12 US disclosed
CN-1922158-A Isothiourea derivatives NOVARTIS AG (CH) 2007-02-28 CN disclosed
EP-1720845-A1 ISOTHIOUREA DERIVATIVES Novartis AG (CH) 2006-11-15 EP disclosed
EP-1669352-A1 THIAZOLINE DERIVATIVE AND USE OF THE SAME Takeda Pharmaceutical Company Limited (JP) 2006-06-14 EP disclosed
WO-2005085219-A1 ISOTHIOUREA DERIVATIVES NOVARTIS AG (CH) 2005-09-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070161618-A1 Isothiourea derivatives TPMT, HLA-DRB1, IRF3 CXCR4 932/4885ALDH1A1 489/4885GAA 2190/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.