SCHEMBL353138

SCHEMBL353138

Cc1nccc(C(N)=O)c1C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT3 Q9NTG7 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
KDM4E B2RXH2 3/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
MKNK1 Q9BUB5 1/20 0.42
MKNK2 Q9HBH9 1/20 0.42
NNMT P40261 4/20 0.42
P2RX7 Q99572 1/20 0.42
PIK3CB P42338 1/20 0.41
NPC1 O15118 1/20 0.39
MAPT P10636 1/20 0.39
AHR P35869 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
PARP1 P09874 3/20 0.39
CDC7 O00311 1/20 0.38
CCNC P24863 1/20 0.37
CDK8 P49336 1/20 0.37
LIMK1 P53667 1/20 0.37
ALDH1A1 P00352 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5796678 0.98 SIRT3 (0.44) SIRT3TDP1KDM4EL3MBTL1MKNK1
SCHEMBL5169967 0.82 NOS3 (0.52) SIRT3TDP1KDM4EL3MBTL1MKNK1
SCHEMBL5169958 0.82 SIRT3 (0.44) SIRT3TDP1KDM4EL3MBTL1MKNK1
SCHEMBL19439221 0.82 SIRT3 (0.44) SIRT3TDP1KDM4EL3MBTL1MKNK2
SCHEMBL9002808 0.82 SIRT3 (0.44) SIRT3TDP1KDM4EL3MBTL1MKNK1
SCHEMBL6628065 0.81 SMN1; SMN2 (0.45) KDM4EP2RX7RAB9ASMN1; SMN2ALDH1A1
SCHEMBL353106 0.81 KDM4E (0.47) TDP1KDM4EL3MBTL1MAPTRAB9A
SCHEMBL16447580 0.80 SIRT3 (0.43) SIRT3TDP1KDM4EL3MBTL1MKNK1
SCHEMBL15991433 0.80 SIRT3 (0.43) SIRT3TDP1KDM4EL3MBTL1NNMT
SCHEMBL17195496 0.80 MKNK1 (0.44) SIRT3TDP1KDM4EL3MBTL1MKNK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 119 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111868037-A Fused cyclic urea derivatives as CRHR2 antagonists 拉夸里亚创药株式会社 2020-10-30 CN claimed
CN-101065358-B 3-arylamino pyridine derivatives MERCK SERONO SA 2015-03-11 CN claimed
CN-103408486-A Preparation method of 4-pyridinemethanol UNIV GUILIN TECH GUT 2013-11-27 CN claimed
EP-1802579-B1 Derivatives of 3-arylaminopyridine MERCK SERONO SA (CH) 2013-11-20 EP claimed
CN-103249721-A Arylamine Derivatives as TTX-S Blockers RAQUALIA PHARMA INC 2013-08-14 CN claimed
CN-101065358-A 3-arylamino pyridine derivatives APPLIED RESEARCH SYSTEMS (AN) 2007-10-31 CN claimed
WO-1998033786-A9 ACCELERATED CATALYSIS OF OLEFINIC EPOXIDATIONS 1998-12-30 WO claimed
WO-1998033786-A1 ACCELERATED CATALYSIS OF OLEFINIC EPOXIDATIONS THE SCRIPPS RESEARCH INSTITUTE (US) 1998-08-06 WO claimed
US-20250129044-A1 PYRIDINYL DERIVATIVES AS SODIUM CHANNEL ACTIVATORS XENON PHARMACEUTICALS INC. (CA) 2025-04-24 US disclosed
CN-113307772-B Human plasma kallikrein inhibitors 拜奥克里斯特制药公司 2024-06-28 CN disclosed
CN-118103369-A Pyridolactam derivatives, preparation method and application thereof 浙江海正药业股份有限公司 2024-05-28 CN disclosed
CN-112312905-B Tetrazole-containing inhibitors of apoptosis signal-regulating kinase 1 and methods of use thereof 英安塔制药有限公司 2024-03-15 CN disclosed
CN-117355303-A Compounds and their use for the treatment of neurodegenerative, degenerative and metabolic disorders 佛罗里达大学研究基金会公司 2024-01-05 CN disclosed
CN-117105933-A Substituted 6-azabenzimidazole compounds having HPK1 inhibitory activity 吉利德科学公司 2023-11-24 CN disclosed
CN-1390215-A Tyrosine kinase inhibitors MERCK & CO INC (US) 2003-01-08 CN disclosed
CN-1320652-A Salt of polyacylimino-amic acid and polyacylimine film formed therefrom PLEX TECHNOLOGIES CORP (US) 2001-11-07 CN disclosed
WO-1998033786-A9 ACCELERATED CATALYSIS OF OLEFINIC EPOXIDATIONS 1998-12-30 WO disclosed
WO-1998033786-A1 ACCELERATED CATALYSIS OF OLEFINIC EPOXIDATIONS THE SCRIPPS RESEARCH INSTITUTE (US) 1998-08-06 WO disclosed
CN-1184813-A Pyridine derivatives, process for preparing the same, and intermediate therefor TANABE SEIYAKU CO (JP) 1998-06-17 CN disclosed
US-4693726-A Process for dyeing or printing cellulose fibers or cellulose blend fibers with pyridinium-triazine reactive dye, axable without alkali HOECHST AKTIENGESELLSCHAFT (DE) 1987-09-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250129044-A1 PYRIDINYL DERIVATIVES AS SODIUM CHANNEL ACTIVATORS SCN1B, SCN1A, SCN2B SIRT3 760/4885TDP1 1890/4885KDM4E 1340/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.