SCHEMBL3535268

SCHEMBL3535268

CCN1CCCC1C(C)N

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.38
HTT P42858 1/20 0.36
ALDH1A1 P00352 1/20 0.33
DPP4 P27487 6/20 0.33
DPP8 Q6V1X1 3/20 0.33
DPP9 Q86TI2 3/20 0.33
DPP7 Q9UHL4 3/20 0.33
FAP Q12884 2/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4038087 1.00 L3MBTL1 (0.38) L3MBTL1HTTALDH1A1DPP4DPP8
SCHEMBL4035789 1.00 L3MBTL1 (0.38) L3MBTL1HTTALDH1A1DPP4DPP8
Ammonia Solution, Strong SCHEMBL9243093 0.98 L3MBTL1 (0.37) L3MBTL1HTTALDH1A1DPP4DPP8
SCHEMBL4202492 0.85 L3MBTL1 (0.36) L3MBTL1HTTALDH1A1DPP4DPP8
SCHEMBL12299850 0.83 L3MBTL1 (0.40) L3MBTL1HTTALDH1A1KMT2A
SCHEMBL12658782 0.83 L3MBTL1 (0.40) L3MBTL1HTTALDH1A1KMT2A
SCHEMBL12658780 0.83 L3MBTL1 (0.40) L3MBTL1HTTALDH1A1KMT2A
SCHEMBL23372707 0.79 L3MBTL1 (0.38) L3MBTL1HTTALDH1A1KMT2A
SCHEMBL21959058 0.79 HTT (0.39) L3MBTL1HTTALDH1A1KMT2A
SCHEMBL31474253 0.79 L3MBTL1 (0.41) L3MBTL1HTTALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021022163-A2 COMPOUNDS AND USES THEREOF FOGHORN THERAPEUTICS INC. (US) 2021-02-04 WO disclosed
US-10874640-B2 Substituted pyrrolizine compounds and uses thereof GILEAD SCIENCES, INC. (US) 2020-12-29 US disclosed
US-20200061024-A1 SUBSTITUTED PYRROLIZINE COMPOUNDS AND USES THEREOF GILEAD SCIENCES, INC. 2020-02-27 US disclosed
US-7709479-B1 Quinazoline derivatives and their use as pharmaceuticals ASTRAZENECA (SE) 2010-05-04 US disclosed
US-20080058365-A1 Fused heterocyclic compounds AMGEN INC. 2008-03-06 US disclosed
US-7253179-B2 Fused heterocyclic compounds AMGEN INC. (US) 2007-08-07 US disclosed
US-20040147538-A1 Fused heterocyclic compounds AMGEN INC. 2004-07-29 US disclosed
US-6515122-B1 The invention further relates to combinatorial libraries containing two or more such compounds, as well as methods of preparing tetracyclic benzimidazole derivative compounds. LION BIOSCIENCE AG (DE) 2003-02-04 US disclosed
EP-0604895-A1 Pigment compounds SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1994-07-06 EP disclosed
US-5317015-A Azacyclic bisphosphonates as anticholesterolemic agents RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1994-05-31 US disclosed
EP-0273401-B1 ISOINDOLIN-1-ONE DERIVATIVE AND ANTIARRHYTHMIC AGENT KYOWA HAKKO KOGYO KABUSHIKI KAISHA (JP) 1992-11-11 EP disclosed
US-4849441-A Isoindolin-1-one derivative and antiarrhythmic agent KYOWA HAKKO KOGYO CO., LTD. (JP) 1989-07-18 US disclosed
US-4772600-A MUSCLE RELAXANTS, ANTICONVULSANTS, ANXIOLYTIC A. H. ROBINS COMPANY, INC. (US) 1988-09-20 US disclosed
EP-0000977-B1 AGGREGATED POLYELECTROLYTES, THEIR PREPARATION AND USES IN THE FRACTIONATION OF BLOOD AND OTHER PROTEINACEOUS SUBSTANCES MONSANTO COMPANY (US) 1981-09-02 EP disclosed
US-4118554-A HEATING IN INERT ORGANIC SOLVENT, CONTAINS AMINE-IMIDE FUNCTIONAL GROUPS MONSANTO COMPANY (US) 1978-10-03 US disclosed
US-4097473-A ADSORPTION ON ETHYLENE-MALEIC ANHYDRIDE COPOLYMER CONTAINING PENDANT DIMETHYLAMINOPROPYL FUNCTIONAL GROUPS MONSANTO COMPANY (US) 1978-06-27 US disclosed
US-3959477-A Methods of protection against emesis in mammals by administration of a heterocyclic benzamide SOCIETE D'ETUDES SCIENTIFIQUES ET INDUSTRIELLES DE L'ILE-DE-FRANCE (FR) 1976-05-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200061024-A1 SUBSTITUTED PYRROLIZINE COMPOUNDS AND USES THEREOF HMBS, DHFR, HCCS L3MBTL1 4026/4885HTT 1814/4885ALDH1A1 4332/4885
US-10874640-B2 Substituted pyrrolizine compounds and uses thereof HMBS, DHFR, HCCS L3MBTL1 4026/4885HTT 1814/4885ALDH1A1 4332/4885
US-20080058365-A1 Fused heterocyclic compounds GIPR, MC4R, GPR119 L3MBTL1 3838/4885HTT 396/4885ALDH1A1 1509/4885
US-20040147538-A1 Fused heterocyclic compounds GIPR, MC4R, GPR119 L3MBTL1 3838/4885HTT 396/4885ALDH1A1 1509/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.