SCHEMBL3538485

SCHEMBL3538485

Fc1ccc2[nH]nc(-c3nc4cc(Cl)ccc4[nH]3)c2c1

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 8/20 0.51
FGFR1 P11362 4/20 0.50
ITK Q08881 2/20 0.49
FLT1 P17948 1/20 0.49
FLT3 P36888 2/20 0.46
FADS1 O60427 1/20 0.44
CLK4 Q9HAZ1 1/20 0.43
HTR2A P28223 1/20 0.42
CHEK1 O14757 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3538345 0.84 PDPK1 (0.72) PDPK1FGFR1ITKFLT1FLT3
SCHEMBL3537973 0.84 PDPK1 (0.51) PDPK1FGFR1ITKFLT1FLT3
SCHEMBL3533017 0.84 PDPK1 (0.71) PDPK1FGFR1ITKFLT1FLT3
SCHEMBL5953085 0.83 FGFR1 (0.51) PDPK1FGFR1ITKFLT1FLT3
SCHEMBL3532319 0.82 PDPK1 (0.51) PDPK1FGFR1ITKFLT1FLT3
SCHEMBL3531870 0.81 PDPK1 (0.71) PDPK1FGFR1ITKFLT1FLT3
SCHEMBL3542692 0.81 PDPK1 (0.56) PDPK1FGFR1ITKFLT1FLT3
SCHEMBL5951667 0.80 MAP3K8 (0.51) PDPK1FGFR1ITKFLT1FLT3
SCHEMBL3534190 0.79 MAPT (0.55) PDPK1FGFR1FLT1
SCHEMBL3538807 0.79 ALDH1A1 (0.58) PDPK1FGFR1ITKFLT1FLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7642278-B2 Nitrogen compounds such as 3-(5-morpholin-4-yl-1H-benz-imidazol-2-yl)-1H-indazole and/or isomers, used as immunology modulators, antidiabetic agents, antiogenesis inhibitors or for prophylaxis of Alzheimer's disease NOVARTIS VACCINES AND DIAGNOSTICS, INC. (US) 2010-01-05 US disclosed
US-7064215-B2 Indazole benzimidazole compounds CHIRON CORPORATION (US) 2006-06-20 US disclosed
US-20060079564-A1 Indazole benzimidazole compounds CHIRON CORPORATION 2006-04-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060079564-A1 Indazole benzimidazole compounds ABL1, ABL2, ALK PDPK1 1862/4885FGFR1 886/4885ITK 1055/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.