SCHEMBL3548022

SCHEMBL3548022

CN1CC[C@@H](N)[C@@H]1Cc1ccsc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.44
MEN1 O00255 1/20 0.44
KDM4A O75164 1/20 0.44
MAPT P10636 1/20 0.44
KMT2A Q03164 1/20 0.44
HSD17B10 Q99714 1/20 0.44
KDM4C Q9H3R0 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
TAAR1 Q96RJ0 1/20 0.36
LTA4H P09960 1/20 0.35
LMNA P02545 2/20 0.35
SIGMAR1 Q99720 2/20 0.34
OPRM1 P35372 4/20 0.33
OPRD1 P41143 4/20 0.33
OPRK1 P41145 4/20 0.33
DPP4 P27487 1/20 0.33
DPP8 Q6V1X1 1/20 0.33
DPP9 Q86TI2 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28241887 0.78 PRMT6 (0.45) SIGMAR1OPRM1OPRD1OPRK1
SCHEMBL3551226 0.78 PRMT6 (0.45) SIGMAR1OPRM1OPRD1OPRK1
SCHEMBL3550203 0.75 ALDH1A1 (0.41) ALDH1A1L3MBTL1
SCHEMBL13344520 0.73 NR1I2 (0.40) ALDH1A1MEN1KDM4AMAPTKMT2A
SCHEMBL13369098 0.73 NR1I2 (0.40) ALDH1A1MEN1KDM4AMAPTKMT2A
SCHEMBL3548008 0.71 ACHE (0.47) KMT2ASIGMAR1DPP4CYP1A2
SCHEMBL3548356 0.71 HSD17B2 (0.47) ALDH1A1MAPTL3MBTL1TAAR1SIGMAR1
SCHEMBL3551208 0.71 SLC6A3 (0.43) ALDH1A1SIGMAR1
SCHEMBL3550805 0.67 CXCR4 (0.43) ALDH1A1MEN1MAPTKMT2ATAAR1
SCHEMBL5146706 0.67 CXCR4 (0.43) ALDH1A1MEN1MAPTKMT2ATAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7714021-B2 Pyrrolidin-3-yl compounds useful as beta-secretase inhibitors for the treatment of Alzheimer's disease MERCK & CO., INC. (US) 2010-05-11 US disclosed
US-20080287523-A1 Pyrrolidin-3-Yl Compounds Useful as Beta-Secretase Inhibitors for the Treatment of Alzheimer's Disease MERCK SHARP & DOHME LLC 2008-11-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080287523-A1 Pyrrolidin-3-Yl Compounds Useful as Beta-Secretase Inhibitors for the Treatment of Alzheimer's Disease BACE1, BACE2, APP ALDH1A1 2813/4885MEN1 3555/4885KDM4A 1646/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.