SCHEMBL3552039

SCHEMBL3552039

COC(=O)c1ccc(N2CCN(c3ccc(C(C)(C)C)cc3)C2=O)cc1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.50
CA2 P00918 2/20 0.50
ALDH1A1 P00352 5/20 0.47
HTT P42858 2/20 0.46
KDM4E B2RXH2 1/20 0.46
MAPT P10636 3/20 0.45
DRD2 P14416 1/20 0.44
DRD3 P35462 1/20 0.44
KCNH2 Q12809 1/20 0.44
EGFR P00533 1/20 0.44
HDAC1 Q13547 3/20 0.44
LMNA P02545 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
CTSG P08311 1/20 0.43
CMA1 P23946 1/20 0.43
GRIN2B Q13224 1/20 0.43
GAA P10253 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3555407 0.87 CTSG (0.44) ALDH1A1MAPTEGFRHDAC1SMN1; SMN2
SCHEMBL3550945 0.87 HDAC1 (0.63) CA1CA2ALDH1A1DRD2DRD3
SCHEMBL592406 0.81 CA1 (0.68) CA1CA2ALDH1A1MAPTEGFR
SCHEMBL3553014 0.80 EGFR (0.52) ALDH1A1KDM4EMAPTEGFRHDAC1
Water SCHEMBL28249729 0.79 CA1 (0.66) CA1CA2ALDH1A1MAPTEGFR
SCHEMBL14686979 0.78 ALDH1A1 (0.48) CA1CA2ALDH1A1HTTMAPT
SCHEMBL3561479 0.78 DRD2 (0.48) MAPTDRD2DRD3KCNH2HDAC1
SCHEMBL7716263 0.77 PDE4A (0.46) CA1CA2ALDH1A1HTTMAPT
SCHEMBL3559417 0.77 HDAC1 (0.51) CA1CA2ALDH1A1HTTMAPT
SCHEMBL13006962 0.77 ALDH1A1 (0.56) ALDH1A1KDM4EMAPTDRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100317649-A1 S1P Receptor Modulating Compounds and Use Thereof EPIX PHARMACEUTICALS, INC. (US) 2010-12-16 US disclosed
US-20100317649-A1 S1P Receptor Modulating Compounds and Use Thereof EPIX PHARMACEUTICALS, INC. (US) 2010-12-16 US disclosed
US-7790707-B2 S1P receptor modulating compounds and use thereof EPIX PHARMACEUTICALS INC. (US) 2010-09-07 US disclosed
US-7790707-B2 S1P receptor modulating compounds and use thereof EPIX PHARMACEUTICALS INC. (US) 2010-09-07 US disclosed
US-7790707-B2 S1P receptor modulating compounds and use thereof EPIX PHARMACEUTICALS INC. (US) 2010-09-07 US disclosed
EP-2010524-A2 S1P RECEPTOR MODULATING COMPOUNDS Epix Delaware, Inc. (US) 2009-01-07 EP disclosed
US-20080015177-A1 S1P receptor modulating compounds and use thereof AMGEN INC. 2008-01-17 US disclosed
US-20080015177-A1 S1P receptor modulating compounds and use thereof AMGEN INC. 2008-01-17 US disclosed
US-20080015177-A1 S1P receptor modulating compounds and use thereof AMGEN INC. 2008-01-17 US disclosed
WO-2007109330-A2 S1P RECEPTOR MODULATING COMPOUNDS EPIX DELAWARE, INC. (US) 2007-09-27 WO disclosed
WO-2007109330-A2 S1P RECEPTOR MODULATING COMPOUNDS EPIX DELAWARE, INC. (US) 2007-09-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080015177-A1 S1P receptor modulating compounds and use thereof S1PR1, S1PR2, S1PR5 CA1 4741/4885CA2 4057/4885ALDH1A1 3180/4885
US-20100317649-A1 S1P Receptor Modulating Compounds and Use Thereof S1PR1, S1PR2, S1PR5 CA1 4741/4885CA2 4057/4885ALDH1A1 3180/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.