SCHEMBL3562883

SCHEMBL3562883

CC(NCCOC(Cc1ccccc1)C1=COCO1)c1nc(-n2ccnc2)ns1

nearest known ligand 0.39

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 15/20 0.39
NOS1 P29475 11/20 0.36
POLB P06746 1/20 0.33
NPC1 O15118 1/20 0.33
TSHR P16473 1/20 0.33
HSD17B10 Q99714 1/20 0.33
PDE5A O76074 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3569290 0.84 NOS2 (0.57) NOS2NOS1POLBNPC1TSHR
SCHEMBL3564769 0.74 NOS2 (0.37) NOS2NOS1POLBPDE5A
SCHEMBL3559005 0.73 NOS2 (0.38) NOS2NOS1NPC1TSHRHSD17B10
SCHEMBL3620097 0.72 NOS2 (0.41) NOS2NOS1
SCHEMBL3562878 0.72 NOS2 (0.72) NOS2NOS1
SCHEMBL3615118 0.72 TSHR (0.38) NOS2NOS1POLBTSHRHSD17B10
SCHEMBL3566903 0.71 NOS2 (0.50) NOS2NOS1
SCHEMBL3567894 0.70 NOS2 (0.56) NOS2NOS1
SCHEMBL3568583 0.70 NOS2 (0.35) NOS2NOS1NPC1TSHRHSD17B10
SCHEMBL3556926 0.69 NOS2 (0.46) NOS2NOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7825256-B2 Inducible nitric oxide synthase dimerization inhibitors KALYPSYS, INC. (US) 2010-11-02 US disclosed
EP-1817030-A2 INDUCIBLE NITRIC OXIDE SYNTHASE DIMERIZATION INHIBITORS Kalypsys, Inc. (US) 2007-08-15 EP disclosed
WO-2006060424-A2 INDUCIBLE NITRIC OXIDE SYNTHASE DIMERIZATION INHIBITORS KALYPSYS, INC. (US) 2006-06-08 WO disclosed