SCHEMBL3569290

SCHEMBL3569290

Cc1cc(C(C)NCCOC(Cc2ccccc2)C2=COCO2)nc(-n2ccnc2)n1

nearest known ligand 0.57

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 12/20 0.57
NOS1 P29475 3/20 0.51
POLB P06746 1/20 0.33
NPC1 O15118 1/20 0.33
TSHR P16473 1/20 0.33
HSD17B10 Q99714 1/20 0.33
PDE5A O76074 5/20 0.33
TBXAS1 P24557 2/20 0.33
PDE3B Q13370 2/20 0.33
PDE3A Q14432 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3562883 0.84 NOS2 (0.39) NOS2NOS1POLBNPC1TSHR
SCHEMBL3571989 0.82 NOS2 (0.53) NOS2NOS1POLBNPC1TSHR
SCHEMBL3570486 0.73 NOS2 (0.39) NOS2NOS1TSHR
SCHEMBL3559827 0.73 NOS2 (0.44) NOS2NOS1PDE5ATBXAS1PDE3B
SCHEMBL3569287 0.73 NOS2 (1.00) NOS2NOS1
SCHEMBL3566047 0.72 NOS2 (0.39) NOS2NOS1
SCHEMBL3563614 0.72 NOS2 (0.51) NOS2NOS1NPC1TSHRHSD17B10
SCHEMBL3571983 0.71 NOS2 (0.73) NOS2NOS1
SCHEMBL3556345 0.71 NOS2 (0.55) NOS2NOS1
SCHEMBL3561919 0.71 NOS2 (0.54) NOS2NOS1NPC1TSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7825256-B2 Inducible nitric oxide synthase dimerization inhibitors KALYPSYS, INC. (US) 2010-11-02 US disclosed