SCHEMBL3559005

SCHEMBL3559005

CC(NC(CNCc1ccccc1)CC1=COCO1)c1nc(-n2ccnc2)ns1

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 18/20 0.38
NOS1 P29475 15/20 0.38
PDE5A O76074 1/20 0.35
PTGS1 P23219 1/20 0.35
TBXAS1 P24557 1/20 0.35
PTGS2 P35354 1/20 0.35
PDE3B Q13370 1/20 0.35
PDE3A Q14432 1/20 0.35
NPC1 O15118 1/20 0.33
TSHR P16473 1/20 0.33
HSD17B10 Q99714 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3559827 0.84 NOS2 (0.44) NOS2NOS1PDE5APTGS1TBXAS1
SCHEMBL3566770 0.82 ADRB2 (0.32) PDE5APTGS1TBXAS1PTGS2PDE3B
SCHEMBL3559740 0.78 NOS2 (0.46) NOS2NOS1
SCHEMBL3560293 0.76 NOS2 (0.48) NOS2NOS1
Hydrochloric Acid SCHEMBL3563512 0.76 NOS2 (0.48) NOS2NOS1
SCHEMBL3556543 0.75 NOS2 (0.51) NOS2NOS1
SCHEMBL3567376 0.74 NOS2 (0.51) NOS2NOS1
SCHEMBL3562883 0.73 NOS2 (0.39) NOS2NOS1PDE5ANPC1TSHR
SCHEMBL3571843 0.72 NOS2 (0.51) NOS2NOS1
SCHEMBL3570858 0.71 NOS2 (0.55) NOS2NOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7825256-B2 Inducible nitric oxide synthase dimerization inhibitors KALYPSYS, INC. (US) 2010-11-02 US disclosed
US-20060116515-A1 Inducible nitric oxide synthase dimerization inhibitors KALYPSYS, INC. 2006-06-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060116515-A1 Inducible nitric oxide synthase dimerization inhibitors NOS3, NOS2, NOS1 NOS2 2/4885NOS1 3/4885PDE5A 261/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.