SCHEMBL3570650

SCHEMBL3570650

CC(C)(C)c1ccc(CN(CCc2ccc(Cl)c(Cl)c2)C(=O)c2cc(Cl)cnc2NCCO)cc1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CCR9 P51686 8/20 0.41
ESRRG P62508 2/20 0.36
ESRRB O95718 1/20 0.36
NR1I3 Q14994 1/20 0.35
NR1H4 Q96RI1 1/20 0.35
VNN1 O95497 1/20 0.35
CNR1 P21554 1/20 0.34
F10 P00742 1/20 0.34
HSP90AA1 P07900 2/20 0.33
TRPV1 Q8NER1 1/20 0.33
SIGMAR1 Q99720 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3585932 0.91 CCR9 (0.36) CCR9ESRRGESRRBNR1I3NR1H4
SCHEMBL3576692 0.89 ESRRG (0.37) CCR9ESRRGESRRBNR1I3NR1H4
SCHEMBL3581747 0.88 CCR9 (0.39) CCR9ESRRGESRRBNR1I3NR1H4
SCHEMBL3580209 0.85 MCHR1 (0.40) CCR9ESRRGESRRBNR1I3NR1H4
SCHEMBL3581265 0.85 NR1H4 (0.39) CCR9ESRRGESRRBNR1I3NR1H4
SCHEMBL3576645 0.83 HSP90AA1 (0.37) ESRRGESRRBNR1I3NR1H4HSP90AA1
SCHEMBL3583608 0.83 ESRRG (0.35) ESRRGESRRBNR1I3NR1H4HSP90AA1
SCHEMBL3575573 0.83 HSP90AA1 (0.36) ESRRGESRRBNR1I3NR1H4HSP90AA1
SCHEMBL3580374 0.81 ESRRG (0.36) CCR9ESRRGESRRBNR1I3NR1H4
SCHEMBL1397638 0.81 HCRTR1 (0.37) CCR9NR1I3SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7678818-B2 Anthranilamide and 2-amino-heteroarene-carboxamide compounds HOFFMANN-LA ROCHE INC. (US) 2010-03-16 US claimed
EP-1984340-B1 ANTHRANILAMIDE/2-AMINO-HETEROARENE CARBOXAMIDE DERIVATIVES HOFFMANN LA ROCHE (CH) 2012-06-27 EP disclosed