SCHEMBL3580209

SCHEMBL3580209

CC(C)(C)c1ccc(CN(CCc2ccc(Cl)c(Cl)c2)C(=O)c2cc(Cl)cnc2NC2CC2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 3/20 0.40
BTK Q06187 1/20 0.37
HDAC3 O15379 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
ESRRG P62508 2/20 0.34
NR1H4 Q96RI1 1/20 0.34
CCR9 P51686 1/20 0.34
ESRRB O95718 1/20 0.34
CRHR1 P34998 3/20 0.34
MELK Q14680 2/20 0.34
OPRM1 P35372 1/20 0.34
OPRD1 P41143 1/20 0.34
THRB P10828 1/20 0.34
NR1I3 Q14994 1/20 0.33
MEN1 O00255 1/20 0.33
HPGD P15428 1/20 0.33
KMT2A Q03164 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
IRAK4 Q9NWZ3 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3576972 0.92 BTK (0.36) BTKHDAC3HDAC8HDAC6ESRRG
SCHEMBL3579944 0.91 MCHR1 (0.39) MCHR1CRHR1OPRM1OPRD1
SCHEMBL3576692 0.89 ESRRG (0.37) ESRRGNR1H4CCR9ESRRBOPRM1
SCHEMBL3583661 0.88 BTK (0.41) BTKHDAC3HDAC8HDAC6ESRRG
SCHEMBL3586536 0.88 MCHR1 (0.37) MCHR1BTKHDAC3HDAC8HDAC6
SCHEMBL3585932 0.87 CCR9 (0.36) ESRRGNR1H4CCR9ESRRBOPRM1
SCHEMBL3577036 0.86 MCHR1 (0.43) MCHR1OPRM1OPRD1
SCHEMBL3570650 0.85 CCR9 (0.41) ESRRGNR1H4CCR9ESRRBNR1I3
SCHEMBL3572867 0.85 MEN1 (0.38) HDAC3HDAC8HDAC6ESRRGNR1H4
SCHEMBL3581265 0.85 NR1H4 (0.39) ESRRGNR1H4CCR9ESRRBOPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7678818-B2 Anthranilamide and 2-amino-heteroarene-carboxamide compounds HOFFMANN-LA ROCHE INC. (US) 2010-03-16 US claimed
EP-1984340-B1 ANTHRANILAMIDE/2-AMINO-HETEROARENE CARBOXAMIDE DERIVATIVES HOFFMANN LA ROCHE (CH) 2012-06-27 EP disclosed