SCHEMBL3576645

SCHEMBL3576645

CCNc1ncc(C)cc1C(=O)N(CCc1ccc(Cl)c(Cl)c1)Cc1ccc(C(C)(C)C)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 2/20 0.37
GRM5 P41594 1/20 0.36
ESRRG P62508 2/20 0.35
NR1H4 Q96RI1 1/20 0.35
ESRRB O95718 1/20 0.35
OPRM1 P35372 1/20 0.35
OPRD1 P41143 1/20 0.35
NR1I3 Q14994 1/20 0.34
HCRTR1 O43613 1/20 0.33
HCRTR2 O43614 1/20 0.33
RPS6KB1 P23443 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
CETP P11597 1/20 0.33
LMNA P02545 1/20 0.33
GAA P10253 1/20 0.32
HTT P42858 1/20 0.32
GFER P55789 1/20 0.32
IKBKB O14920 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3585932 0.92 CCR9 (0.36) HSP90AA1GRM5ESRRGNR1H4ESRRB
SCHEMBL3580374 0.91 ESRRG (0.36) HSP90AA1GRM5ESRRGNR1H4ESRRB
SCHEMBL3583608 0.90 ESRRG (0.35) HSP90AA1ESRRGNR1H4ESRRBOPRM1
SCHEMBL3575573 0.90 HSP90AA1 (0.36) HSP90AA1ESRRGNR1H4ESRRBOPRM1
SCHEMBL3570650 0.83 CCR9 (0.41) HSP90AA1ESRRGNR1H4ESRRBNR1I3
SCHEMBL3587153 0.83 ESRRG (0.36) HSP90AA1GRM5ESRRGNR1H4ESRRB
SCHEMBL3576692 0.83 ESRRG (0.37) HSP90AA1ESRRGNR1H4ESRRBOPRM1
SCHEMBL3574285 0.81 ESRRG (0.36) HSP90AA1ESRRGNR1H4ESRRBOPRM1
SCHEMBL3577133 0.81 CYP51A1 (0.36) HSP90AA1ESRRGNR1H4ESRRBOPRM1
SCHEMBL3584126 0.81 ESRRG (0.36) HSP90AA1ESRRGNR1H4ESRRBOPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7678818-B2 Anthranilamide and 2-amino-heteroarene-carboxamide compounds HOFFMANN-LA ROCHE INC. (US) 2010-03-16 US claimed
EP-1984340-B1 ANTHRANILAMIDE/2-AMINO-HETEROARENE CARBOXAMIDE DERIVATIVES HOFFMANN LA ROCHE (CH) 2012-06-27 EP disclosed