SCHEMBL3581747

SCHEMBL3581747

CC(C)(C)c1ccc(CN(CCc2ccc(Cl)c(Cl)c2)C(=O)c2cccnc2NCCO)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR9 P51686 4/20 0.39
KDR P35968 1/20 0.37
RAF1 P04049 1/20 0.37
MAP2K1 Q02750 1/20 0.37
ALDH1A1 P00352 2/20 0.36
HPGD P15428 2/20 0.36
KDM4E B2RXH2 1/20 0.36
HSD17B10 Q99714 1/20 0.36
ESRRB O95718 1/20 0.36
ESRRG P62508 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
PDPK1 O15530 1/20 0.35
NR1H4 Q96RI1 1/20 0.35
VNN1 O95497 1/20 0.35
OPRM1 P35372 1/20 0.34
OPRD1 P41143 1/20 0.34
ATM Q13315 1/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3580658 0.89 RAF1 (0.39) KDRRAF1MAP2K1ESRRBESRRG
SCHEMBL3570650 0.88 CCR9 (0.41) CCR9ESRRBESRRGNR1H4VNN1
SCHEMBL3583661 0.85 BTK (0.41) RAF1MAP2K1ESRRBESRRGMEN1
SCHEMBL3573203 0.85 RAF1 (0.40) RAF1MAP2K1ESRRBESRRGMEN1
SCHEMBL3582883 0.84 RAF1 (0.40) RAF1MAP2K1ESRRBESRRGMEN1
SCHEMBL3575452 0.82 KMT2A (0.42) RAF1MAP2K1ALDH1A1ESRRBESRRG
SCHEMBL3580336 0.79 MAPT (0.42) RAF1MAP2K1HSD17B10MEN1KMT2A
SCHEMBL3581464 0.79 TRPV1 (0.41) RAF1MAP2K1HSD17B10MEN1KMT2A
SCHEMBL3585932 0.79 CCR9 (0.36) CCR9ESRRBESRRGNR1H4OPRM1
SCHEMBL3576645 0.78 HSP90AA1 (0.37) ESRRBESRRGNR1H4OPRM1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7678818-B2 Anthranilamide and 2-amino-heteroarene-carboxamide compounds HOFFMANN-LA ROCHE INC. (US) 2010-03-16 US claimed
EP-1984340-B1 ANTHRANILAMIDE/2-AMINO-HETEROARENE CARBOXAMIDE DERIVATIVES HOFFMANN LA ROCHE (CH) 2012-06-27 EP disclosed