SCHEMBL3580122

SCHEMBL3580122

NC(=O)c1cccc2nc(-c3ccc(N4CCN(Cc5ccccc5)CC4)cc3)[nH]c12

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AURKB Q96GD4 3/20 0.56
AURKA O14965 2/20 0.56
KDR P35968 2/20 0.56
PARP1 P09874 8/20 0.52
CHEK2 O96017 3/20 0.51
JAK2 O60674 1/20 0.49
ACHE P22303 1/20 0.47
KDM1A O60341 1/20 0.47
USP2 O75604 1/20 0.46
TP53 P04637 1/20 0.46
ALOX15 P16050 1/20 0.46
TSHR P16473 1/20 0.46
MAPK1 P28482 1/20 0.46
SLC2A1 P11166 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3585487 0.96 PARP1 (0.54) AURKBAURKAKDRPARP1CHEK2
SCHEMBL3578629 0.89 AURKB (0.64) AURKBAURKAKDRPARP1CHEK2
SCHEMBL3582282 0.87 AURKB (0.61) AURKBAURKAKDRPARP1CHEK2
SCHEMBL6805222 0.87 AURKA (0.75) AURKBAURKAKDRPARP1CHEK2
SCHEMBL3580117 0.84 AURKB (0.77) AURKBAURKAKDRPARP1CHEK2
SCHEMBL3574441 0.84 AURKA (0.75) AURKBAURKAPARP1CHEK2ACHE
SCHEMBL6806441 0.84 AURKB (0.70) AURKBAURKAKDRPARP1CHEK2
SCHEMBL3582849 0.83 AURKB (0.58) AURKBAURKAKDRPARP1CHEK2
SCHEMBL3587289 0.83 AURKA (0.56) AURKBAURKAPARP1CHEK2JAK2
SCHEMBL5620766 0.83 AURKA (0.52) AURKBAURKAKDRPARP1JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7781596-B1 Substituted 2-phenylbenzimidazoles, the production thereof and their use ABBOTT LABORATORIES (US) 2010-08-24 US disclosed