SCHEMBL3576126

SCHEMBL3576126

CC(C)(C)c1ccc(CN(CCc2ccc(Cl)c(Cl)c2)C(=O)c2ccncc2N)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 2/20 0.37
ROCK2 O75116 1/20 0.37
CYP51A1 Q16850 2/20 0.37
ESRRG P62508 3/20 0.36
NR1H4 Q96RI1 1/20 0.36
ESRRB O95718 2/20 0.36
OPRM1 P35372 1/20 0.35
OPRD1 P41143 1/20 0.35
TSHR P16473 1/20 0.35
PTGER2 P43116 1/20 0.35
KDM4E B2RXH2 3/20 0.34
ALDH1A1 P00352 3/20 0.34
MEN1 O00255 2/20 0.34
MAPT P10636 2/20 0.34
KMT2A Q03164 2/20 0.34
KDM6B O15054 1/20 0.34
KDM4A O75164 1/20 0.34
THRB P10828 1/20 0.34
KDM4D Q6B0I6 1/20 0.34
KDM4C Q9H3R0 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9957841 0.90 ESRRG (0.39) CYP2C19ROCK2CYP51A1ESRRGNR1H4
SCHEMBL3574429 0.87 KDM4C (0.39) ROCK2CYP51A1ESRRGNR1H4ESRRB
SCHEMBL3571051 0.87 NR1H4 (0.37) ROCK2CYP51A1ESRRGNR1H4ESRRB
SCHEMBL3572359 0.84 TRPV1 (0.37) ROCK2ESRRGNR1H4ESRRBOPRM1
SCHEMBL3577133 0.84 CYP51A1 (0.36) ROCK2CYP51A1ESRRGNR1H4ESRRB
SCHEMBL3582883 0.83 RAF1 (0.40) CYP2C19ESRRGNR1H4ESRRBOPRM1
SCHEMBL3578664 0.82 CYP2C19 (0.39) CYP2C19ESRRGNR1H4ESRRBOPRM1
SCHEMBL3581265 0.81 NR1H4 (0.39) CYP2C19ESRRGNR1H4ESRRBOPRM1
SCHEMBL3573203 0.80 RAF1 (0.40) CYP2C19ESRRGNR1H4ESRRBOPRM1
SCHEMBL9958256 0.80 NR1H4 (0.38) ESRRGNR1H4ESRRBOPRM1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7678818-B2 Anthranilamide and 2-amino-heteroarene-carboxamide compounds HOFFMANN-LA ROCHE INC. (US) 2010-03-16 US claimed
EP-1984340-B1 ANTHRANILAMIDE/2-AMINO-HETEROARENE CARBOXAMIDE DERIVATIVES HOFFMANN LA ROCHE (CH) 2012-06-27 EP disclosed