SCHEMBL3578664

SCHEMBL3578664

Cc1ccc(C(=O)N(CCc2ccc(Cl)c(Cl)c2)Cc2ccc(C(C)(C)C)cc2)c(N)n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 2/20 0.39
NR1H4 Q96RI1 1/20 0.38
ESRRG P62508 2/20 0.37
ESRRB O95718 1/20 0.37
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
MAPT P10636 2/20 0.36
ALDH1A1 P00352 1/20 0.36
TP53 P04637 1/20 0.36
CYP1A2 P05177 1/20 0.36
SIGMAR1 Q99720 1/20 0.36
OPRM1 P35372 1/20 0.35
OPRD1 P41143 1/20 0.35
PSEN1 P49768 1/20 0.35
PSEN2 P49810 1/20 0.35
APH1B Q8WW43 1/20 0.35
NCSTN Q92542 1/20 0.35
APH1A Q96BI3 1/20 0.35
PSENEN Q9NZ42 1/20 0.35
NR1I3 Q14994 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3580712 0.87 NR1H4 (0.39) CYP2C19NR1H4ESRRGESRRBMEN1
SCHEMBL3582883 0.85 RAF1 (0.40) CYP2C19NR1H4ESRRGESRRBMEN1
SCHEMBL3576126 0.82 CYP2C19 (0.37) CYP2C19NR1H4ESRRGESRRBMEN1
SCHEMBL9957841 0.79 ESRRG (0.39) CYP2C19NR1H4ESRRGESRRBMEN1
SCHEMBL3581265 0.78 NR1H4 (0.39) CYP2C19NR1H4ESRRGESRRBMEN1
SCHEMBL3573203 0.78 RAF1 (0.40) CYP2C19NR1H4ESRRGESRRBMEN1
SCHEMBL12521166 0.77 ESRRG (0.44) CYP2C19NR1H4ESRRGESRRBMEN1
SCHEMBL12521072 0.77 TP53 (0.39) NR1H4ESRRGESRRBKMT2AMAPT
SCHEMBL9958256 0.77 NR1H4 (0.38) NR1H4ESRRGESRRBMAPTTP53
SCHEMBL9957773 0.77 NR1H4 (0.38) NR1H4ESRRGESRRBOPRM1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7678818-B2 Anthranilamide and 2-amino-heteroarene-carboxamide compounds HOFFMANN-LA ROCHE INC. (US) 2010-03-16 US claimed
EP-1984340-B1 ANTHRANILAMIDE/2-AMINO-HETEROARENE CARBOXAMIDE DERIVATIVES HOFFMANN LA ROCHE (CH) 2012-06-27 EP disclosed