SCHEMBL3579366

SCHEMBL3579366

CC(C)c1n[nH]c2cnc(NCc3ccccc3)nc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 6/20 0.44
CCNB1 P14635 4/20 0.44
CCNB2 O95067 2/20 0.44
CCNB3 Q8WWL7 2/20 0.44
NPC1 O15118 2/20 0.43
KDM4E B2RXH2 1/20 0.43
MAPT P10636 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
ATM Q13315 1/20 0.41
CDK5 Q00535 5/20 0.41
CDK2 P24941 5/20 0.41
CDK5R1 Q15078 3/20 0.41
CCNT1 O60563 2/20 0.41
CDK9 P50750 2/20 0.41
CCNE1 P24864 2/20 0.41
CDK7 P50613 1/20 0.41
CCNH P51946 1/20 0.41
RAB9A P51151 2/20 0.40
NPSR1 Q6W5P4 1/20 0.40
CDK4 P11802 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3572015 0.82 ALPL (0.47) CDK1CCNB1CCNB2CCNB3NPC1
SCHEMBL3581003 0.80 P2RX3 (0.39) CDK1CCNB1CCNB2CCNB3KDM4E
SCHEMBL3572417 0.79 NTRK1 (0.43) CDK1CDK5CDK2CDK5R1CCNT1
SCHEMBL3574162 0.79 NTRK1 (0.43) CDK1CDK5CDK2CDK5R1CCNT1
SCHEMBL3239170 0.71 CDK1 (0.63) CDK1CCNB1CCNB2CCNB3CDK5
SCHEMBL19117565 0.70 NPC1 (0.61) NPC1RAB9AESR1PDE2AVNN1
SCHEMBL7255577 0.70
SCHEMBL2911505 0.70 NPY5R (0.50) CDK1CCNB1CCNB2CCNB3NPC1
SCHEMBL2912272 0.70 CDK2 (0.51) CDK1CCNB1CCNB2CCNB3NPC1
SCHEMBL2910995 0.70 CDK2 (0.52) CDK1CCNB1CCNB2CCNB3NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7745450-B2 Pyrazolo[4,3-d]pyrimidines, processes for their preparation and methods for therapy INSTITUTE OF EXPERIMENTAL BOTANY (CZ) 2010-06-29 US disclosed
US-20050080097-A1 Pyrazolo[4,3-D]pyrimidines, processes for their preparation and methods for therapy USTAV EXPERIMENTALNI BOTANIKY AV CR (INSTITUTE OF EXPERIMENTAL BOTANY ACADEMY OF 2005-04-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050080097-A1 Pyrazolo[4,3-D]pyrimidines, processes for their preparation and methods for therapy CBR3, DHFR, AKR1C3 CDK1 1081/4885CCNB1 682/4885CCNB2 605/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.