SCHEMBL3580349

SCHEMBL3580349

O=C(C1CC2CCC(C1)N2c1ncccn1)C1(F)C=CC(c2ccccc2)=C(F)C1

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SLC6A7 Q99884 1/20 0.34
KDM4E B2RXH2 3/20 0.33
AGTR2 P50052 1/20 0.31
DPP4 P27487 1/20 0.31
CYP2C19 P33261 1/20 0.30
ALDH1A1 P00352 1/20 0.30
TSHR P16473 1/20 0.30
AOC3 Q16853 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1222089 0.71 THRB (0.30)
SCHEMBL5822729 0.68 KDM4E (0.39) SLC6A7KDM4ECYP2C19ALDH1A1TSHR
SCHEMBL20358219 0.64 RXRA (0.31)
SCHEMBL5822737 0.60 SLC6A7 (0.42) SLC6A7
SCHEMBL3577960 0.60 SLC6A7 (0.41) SLC6A7KDM4ECYP2C19
SCHEMBL3582563 0.60 SLC6A7 (0.52) SLC6A7KDM4EALDH1A1
SCHEMBL28788963 0.60
SCHEMBL1024219 0.60 KDM4E (0.41) SLC6A7KDM4ECYP2C19
SCHEMBL3572446 0.59 SLC6A7 (0.70) SLC6A7
SCHEMBL27587155 0.58 RAB9A (0.33) CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8772291-B2 Multicyclic compounds and methods of their use LEXICON PHARMACEUTICALS, INC. (US) 2014-07-08 US disclosed
US-20100081691-A1 MULTICYCLIC COMPOUNDS AND METHODS OF THEIR USE LEXICON PHARMACEUTICALS, INC. (US) 2010-04-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100081691-A1 MULTICYCLIC COMPOUNDS AND METHODS OF THEIR USE GRIN2C, CHAT, COMT SLC6A7 1113/4885KDM4E 3142/4885AGTR2 1192/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.