SCHEMBL3582780

SCHEMBL3582780

NC(=O)c1cccc2nc(-c3ccc(-n4ccc(CNC(=O)C(F)(F)F)c4)cc3)[nH]c12

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
AURKB Q96GD4 2/20 0.49
KDR P35968 1/20 0.49
PARP1 P09874 16/20 0.38
KCNH2 Q12809 1/20 0.37
MCHR1 Q99705 1/20 0.37
ELANE P08246 1/20 0.35
AURKA O14965 1/20 0.35
DHODH Q02127 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3586255 0.91 KDR (0.41) AURKBKDRPARP1KCNH2MCHR1
SCHEMBL3577370 0.86 KDR (0.65) AURKBKDRPARP1DHODH
SCHEMBL3582143 0.84 AURKB (0.56) AURKBKDRPARP1AURKADHODH
SCHEMBL3580644 0.79 AURKB (0.76) AURKBKDRPARP1AURKADHODH
SCHEMBL3578629 0.79 AURKB (0.64) AURKBKDRPARP1AURKADHODH
SCHEMBL3582340 0.78 AURKB (0.63) AURKBKDRPARP1AURKADHODH
SCHEMBL3586249 0.78 KDR (0.54) AURKBKDRPARP1DHODH
SCHEMBL6580677 0.77 KDR (0.49) AURKBKDRPARP1DHODH
SCHEMBL3581925 0.77 AURKB (0.47) AURKBKDRPARP1AURKADHODH
SCHEMBL3580139 0.75 AURKB (0.46) AURKBKDRPARP1DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7781596-B1 Substituted 2-phenylbenzimidazoles, the production thereof and their use ABBOTT LABORATORIES (US) 2010-08-24 US disclosed