SCHEMBL3584970

SCHEMBL3584970

Cc1cc(N2CCNCC2)ccc1-c1nc2c(C(N)=O)cccc2[nH]1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 18/20 0.53
AURKB Q96GD4 2/20 0.52
AURKA O14965 1/20 0.52
DYRK3 O43781 1/20 0.49
PRKD3 O94806 1/20 0.49
MAP4K4 O95819 1/20 0.49
INSR P06213 1/20 0.49
CSF1R P07333 1/20 0.49
PIM1 P11309 1/20 0.49
CLK2 P49760 1/20 0.49
IRAK1 P51617 1/20 0.49
PRKCD Q05655 1/20 0.49
MAP4K2 Q12851 1/20 0.49
DYRK1A Q13627 1/20 0.49
MELK Q14680 1/20 0.49
MINK1 Q8N4C8 1/20 0.49
PRKD2 Q9BZL6 1/20 0.49
CLK4 Q9HAZ1 1/20 0.49
IRAK4 Q9NWZ3 1/20 0.49
ALK Q9UM73 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6582942 0.85 PARP1 (0.43) PARP1AURKBAURKAPRKD3MAP4K4
SCHEMBL3584976 0.84 ACVR1 (0.42) PARP1AURKBAURKAPIM1CLK4
SCHEMBL3582857 0.83 PARP1 (0.66) PARP1AURKBDYRK3PRKD3MAP4K4
SCHEMBL3580352 0.83 AURKB (0.68) PARP1AURKBAURKADYRK3PRKD3
SCHEMBL7762888 0.82 PDE7A (0.41) PARP1AURKBPRKD3MAP4K4PIM1
SCHEMBL3582368 0.82 AURKB (0.64) PARP1AURKBAURKADYRK3PRKD3
SCHEMBL29411925 0.77 PARP1 (0.72) PARP1AURKBDYRK3PRKD3MAP4K4
SCHEMBL5621808 0.76 PARP1 (0.72) PARP1PARP2
SCHEMBL5621907 0.74 PARP1 (0.66) PARP1
SCHEMBL1741562 0.74 ADRB1 (0.61)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7781596-B1 Substituted 2-phenylbenzimidazoles, the production thereof and their use ABBOTT LABORATORIES (US) 2010-08-24 US disclosed