SCHEMBL3582864

SCHEMBL3582864

NC(=O)c1cccc2nc(-c3cccc(N4CCNCC4)c3)[nH]c12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRK6 P43250 1/20 0.48
HTR7 P34969 7/20 0.46
HTR1A P08908 6/20 0.46
JAK2 O60674 1/20 0.46
CHEK2 O96017 2/20 0.44
PARP1 P09874 4/20 0.43
NPBWR1 P48145 1/20 0.42
PRKCI P41743 2/20 0.42
HTR3E A5X5Y0 1/20 0.41
HTR3B O95264 1/20 0.41
TP53 P04637 1/20 0.41
CYP1A2 P05177 1/20 0.41
ADRB1 P08588 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
THRB P10828 1/20 0.41
CYP2C9 P11712 1/20 0.41
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
SLC6A4 P31645 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3580358 0.89 PARP1 (0.53) JAK2CHEK2PARP1
SCHEMBL3582373 0.85 PARP1 (0.49) CHEK2PARP1
SCHEMBL3584976 0.83 ACVR1 (0.42) HTR7HTR1AJAK2CHEK2PARP1
SCHEMBL3582857 0.83 PARP1 (0.66) CHEK2PARP1
SCHEMBL6805728 0.81 AURKA (0.53) JAK2PARP1
SCHEMBL3585144 0.80 PARP1 (0.64) PARP1TP53HTT
SCHEMBL5621810 0.79 HTR3A (0.52) PARP1HTR3A
SCHEMBL6812407 0.78 AURKA (0.50) JAK2PARP1
SCHEMBL3579908 0.77 PARP1 (0.61) CHEK2PARP1
SCHEMBL3587289 0.77 AURKA (0.56) JAK2CHEK2PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7781596-B1 Substituted 2-phenylbenzimidazoles, the production thereof and their use ABBOTT LABORATORIES (US) 2010-08-24 US disclosed