SCHEMBL3580358

SCHEMBL3580358

NC(=O)c1cccc2nc(-c3ccc(N4CCNCC4)cc3)[nH]c12

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.53
AURKA O14965 1/20 0.50
AURKB Q96GD4 1/20 0.50
CHEK2 O96017 7/20 0.49
PARP2 Q9UGN5 1/20 0.44
ACVR1 Q04771 5/20 0.44
PIM1 P11309 1/20 0.44
PIM3 Q86V86 1/20 0.44
PIM2 Q9P1W9 1/20 0.44
BMPR1B O00238 1/20 0.43
BMPR1A P36894 1/20 0.43
ACVR1B P36896 1/20 0.43
ACVRL1 P37023 1/20 0.43
JAK2 O60674 1/20 0.43
TGFBR1 P36897 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3582373 0.96 PARP1 (0.49) PARP1AURKAAURKBCHEK2PARP2
SCHEMBL3582864 0.89 GRK6 (0.48) PARP1CHEK2JAK2
SCHEMBL3587289 0.88 AURKA (0.56) PARP1AURKAAURKBCHEK2PARP2
SCHEMBL6805728 0.85 AURKA (0.53) PARP1AURKAAURKBJAK2
SCHEMBL3582282 0.85 AURKB (0.61) PARP1AURKAAURKBCHEK2
SCHEMBL3576982 0.85 AURKA (0.52) PARP1AURKAAURKBCHEK2PARP2
SCHEMBL3577227 0.84 AURKA (0.53) PARP1AURKAAURKBCHEK2PARP2
SCHEMBL3584976 0.83 ACVR1 (0.42) PARP1AURKAAURKBCHEK2ACVR1
SCHEMBL3635480 0.83 AURKB (0.56) PARP1AURKAAURKBCHEK2PARP2
SCHEMBL3584716 0.82 AURKB (0.47) PARP1AURKAAURKBCHEK2PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7781596-B1 Substituted 2-phenylbenzimidazoles, the production thereof and their use ABBOTT LABORATORIES (US) 2010-08-24 US disclosed