SCHEMBL3584969

SCHEMBL3584969

CN1CCN(Cc2ccc(B(O)OC(C)(C)C(C)(C)O)cc2)CC1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.47
LMNA P02545 1/20 0.47
MC4R P32245 1/20 0.45
CHKA P35790 6/20 0.44
HDAC6 Q9UBN7 1/20 0.43
KDM4E B2RXH2 2/20 0.43
CA2 P00918 1/20 0.43
NCF1 P14598 1/20 0.43
PRMT6 Q96LA8 1/20 0.43
MAPT P10636 1/20 0.43
NPC1 O15118 2/20 0.42
TP53 P04637 2/20 0.42
RAB9A P51151 2/20 0.42
HPGD P15428 1/20 0.41
HRH3 Q9Y5N1 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17159943 0.95 CHKA (0.53) ALDH1A1LMNACHKAKDM4ECA2
SCHEMBL18580511 0.90 ALDH1A1 (0.48) ALDH1A1LMNAMC4RCHKANPC1
SCHEMBL18580284 0.88 SIGMAR1 (0.42) HRH3
SCHEMBL20635708 0.87 ALDH1A1 (0.47) ALDH1A1LMNAMC4RCHKAHDAC6
SCHEMBL13277275 0.86 SMN1; SMN2 (0.49) ALDH1A1LMNAKDM4EMAPTNPC1
SCHEMBL2509532 0.85 MC4R (0.44) ALDH1A1LMNAMC4RCHKAHDAC6
Hydrochloric Acid SCHEMBL3619140 0.85 SMN1; SMN2 (0.48) KDM4ENPC1TP53RAB9AHPGD
SCHEMBL18580590 0.82 HRH3 (0.35) HDAC6HRH3
SCHEMBL28440571 0.82 LMNA (0.53) ALDH1A1LMNAMC4RCHKAHDAC6
SCHEMBL1428193 0.80 GAA (0.42) ALDH1A1LMNACHKAKDM4ENCF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 43 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12378224-B2 Heteroaryl compounds and their use as Mer inhibitors DONG-A SOCIO HOLDINGS CO., LTD. (KR) 2025-08-05 US disclosed
US-12195446-B2 Heteroaryl compounds and their use as therapeutic drugs DONG-A SOCIO HOLDINGS CO., LTD. (KR) 2025-01-14 US disclosed
US-20230002353-A1 HETEROARYL COMPOUNDS AND THEIR USE AS THERAPEUTIC DRUGS DONG A SOCIO HOLDINGS CO LTD (KR) 2023-01-05 US disclosed
EP-3523292-B1 HETEROARYL COMPOUNDS AND THEIR USE AS MER INHIBITORS DONG A SOCIO HOLDINGS CO LTD (KR) 2021-12-15 EP disclosed
US-20210371398-A1 HETEROARYL COMPOUNDS AND THEIR USE AS MER INHIBITORS DONG A SOCIO HOLDINGS CO LTD (KR) 2021-12-02 US disclosed
US-10947215-B2 Heteroaryl compounds and their use as therapeutic drugs DONG-A SOCIO HOLDINGS CO., LTD. (KR) 2021-03-16 US disclosed
US-10913730-B2 Heteroaryl compounds and their use as Mer inhibitors DONG-A SOCIO HOLDINGS CO., LTD. (KR) 2021-02-09 US disclosed
EP-3344613-B1 HETEROARYL COMPOUNDS AND THEIR USE AS THERAPEUTIC DRUGS DONG A SOCIO HOLDINGS CO LTD (KR) 2020-03-04 EP disclosed
US-20190315716-A1 HETEROARYL COMPOUNDS AND THEIR USE AS MER INHIBITORS DONG-A ST CO., LTD. (KR) 2019-10-17 US disclosed
EP-3523292-A1 HETEROARYL COMPOUNDS AND THEIR USE AS MER INHIBITORS Dong-A Socio Holdings Co., Ltd. (KR) 2019-08-14 EP disclosed
EP-2121687-B1 TRICYCLIC AMINE DERIVATIVES AS PROTEIN TYROSINE KINASE INHIBITORS ASTEX THERAPEUTICS LTD (GB) 2015-10-14 EP disclosed
US-20140275006-A1 AZOLE DERIVATIVE TAISHO PHARMACEUTICAL CO., LTD (JP) 2014-09-18 US disclosed
EP-2772482-A1 AZOLE DERIVATIVE Taisho Pharmaceutical Co., Ltd. (JP) 2014-09-03 EP disclosed
US-20140243315-A1 PYRROLOPYRIMIDINE COMPOUNDS FOR THE TREATMENT OF CANCER THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 2014-08-28 US disclosed
EP-2763988-A1 PYRROLOPYRIMIDINE COMPOUNDS FOR THE TREATMENT OF CANCER The University of North Carolina at Chapel Hill (US) 2014-08-13 EP disclosed
US-8513276-B2 Imidazo[1,2-a]pyridine compounds for use in treating cancer ASTEX THERAPEUTICS LIMITED (GB) 2013-08-20 US disclosed
WO-2013052417-A1 PYRROLOPYRIMIDINE COMPOUNDS FOR THE TREATMENT OF CANCER THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 2013-04-11 WO disclosed
US-20100093718-A1 Compounds ASTEX THERAPEUTICS LIMITED (GB) 2010-04-15 US disclosed
EP-2121687-A2 TRICYCLIC AMINE DERIVATIVES AS PROTEIN TYROSINE KINASE INHIBITORS Astex Therapeutics Limited (GB) 2009-11-25 EP disclosed
WO-2008078100-A2 TRICYCLIC AMINE DERIVATIVES AS PROTEIN TYROSINE KINASE INHIBITORS ASTEX THERAPEUTICS LIMITED (GB) 2008-07-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (10 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10913730-B2 Heteroaryl compounds and their use as Mer inhibitors MERTK, RET, ERBB4 ALDH1A1 3880/4885LMNA 1281/4885MC4R 94/4885
US-10947215-B2 Heteroaryl compounds and their use as therapeutic drugs MERTK, ERBB2, SRC ALDH1A1 3115/4885LMNA 3611/4885MC4R 509/4885
US-12378224-B2 Heteroaryl compounds and their use as Mer inhibitors MERTK, RET, ERBB2 ALDH1A1 3864/4885LMNA 1144/4885MC4R 180/4885
US-12195446-B2 Heteroaryl compounds and their use as therapeutic drugs MERTK, ERBB2, SRC ALDH1A1 3115/4885LMNA 3611/4885MC4R 509/4885
US-20190315716-A1 HETEROARYL COMPOUNDS AND THEIR USE AS MER INHIBITORS MERTK, RET, ERBB4 ALDH1A1 3880/4885LMNA 1281/4885MC4R 94/4885
US-20210371398-A1 HETEROARYL COMPOUNDS AND THEIR USE AS MER INHIBITORS MERTK, RET, ERBB2 ALDH1A1 3864/4885LMNA 1144/4885MC4R 180/4885
US-20140243315-A1 PYRROLOPYRIMIDINE COMPOUNDS FOR THE TREATMENT OF CANCER MERTK, BCR, RET ALDH1A1 2238/4885LMNA 4458/4885MC4R 2828/4885
US-20230002353-A1 HETEROARYL COMPOUNDS AND THEIR USE AS THERAPEUTIC DRUGS MERTK, ERBB2, SRC ALDH1A1 3115/4885LMNA 3611/4885MC4R 509/4885
US-20140275006-A1 AZOLE DERIVATIVE AVPR1B, AVPR1A, AVPR2 ALDH1A1 1469/4885LMNA 4563/4885MC4R 5/4885
US-20100093718-A1 Compounds FGFR1, FGFR2, PDGFRB ALDH1A1 379/4885LMNA 3496/4885MC4R 2284/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.