SCHEMBL3586450

SCHEMBL3586450

NCCCc1c(-c2ccc(Cl)cc2Cl)ncn1CCc1cccc(Cl)c1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 2/20 0.42
HTR6 P50406 1/20 0.38
DPP4 P27487 4/20 0.38
DPP8 Q6V1X1 2/20 0.38
CXCR2 P25025 2/20 0.36
CNR1 P21554 1/20 0.36
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
PNMT P11086 1/20 0.35
BACE1 P56817 1/20 0.34
MAOB P27338 1/20 0.34
GLA P06280 1/20 0.34
HTT P42858 1/20 0.34
UBE2N P61088 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
KDM4C Q9H3R0 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3596861 0.93 TAAR1 (0.47) TAAR1HTR6DPP4DPP8CXCR2
SCHEMBL3586864 0.90 DPP4 (0.45) TAAR1HTR6DPP4DPP8CXCR2
SCHEMBL3604583 0.85 CNR1 (0.41) TAAR1DPP4DPP8CNR1KDM4C
SCHEMBL3604955 0.82 DPP4 (0.48) DPP4DPP8CXCR2CNR1HTT
SCHEMBL3600802 0.79 DPP4 (0.44) DPP4DPP8CXCR2CNR1
SCHEMBL3595338 0.79 PNMT (0.41) TAAR1HTR6DPP4DPP8CXCR2
SCHEMBL3600855 0.78 DPP4 (0.45) DPP4DPP8KDM4C
SCHEMBL3585733 0.78 DPP4 (0.46) DPP4DPP8CXCR2CNR1SMN1; SMN2
SCHEMBL3596995 0.78 SLC6A4 (0.41) DPP4DPP8LMNAMAPT
SCHEMBL3583003 0.77 DPP4 (0.42) DPP4DPP8CXCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728146-B2 Enzyme inhibitors PROBIODRUG AG (DE) 2010-06-01 US claimed