SCHEMBL359363

SCHEMBL359363

NC1CCN(C2=CCCC=N2)CC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.38
HTR3E A5X5Y0 1/20 0.38
MEN1 O00255 1/20 0.38
HTR3B O95264 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
ALOX15 P16050 1/20 0.38
TSHR P16473 1/20 0.38
NFKB1 P19838 1/20 0.38
HTR3A P46098 1/20 0.38
KMT2A Q03164 1/20 0.38
HTR3D Q70Z44 1/20 0.38
HTR3C Q8WXA8 1/20 0.38
AKT2 P31751 5/20 0.34
SSTR2 P30874 1/20 0.34
KIT P10721 1/20 0.34
GSK3B P49841 1/20 0.34
HRH4 Q9H3N8 5/20 0.34
IDH2 P48735 1/20 0.33
CKS1B P61024 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21122995 0.83 LMNA (0.34) MEN1KMT2AIDH2
SCHEMBL8151248 0.68 CASP6 (0.42) MEN1CYP1A2KMT2ACKS1BSKP1
SCHEMBL10055159 0.63 TSHR (0.46) HRH3HTR3EMEN1HTR3BCYP1A2
SCHEMBL13419067 0.61 CYP3A4 (0.63) HRH3HTR3EMEN1HTR3BCYP1A2
SCHEMBL2070684 0.61 KDM4E (0.56) HRH3HTR3EMEN1HTR3BCYP1A2
SCHEMBL6320619 0.60 KDM1A (0.36) HRH3HTR3EMEN1HTR3BCYP1A2
Hydrochloric Acid SCHEMBL5219864 0.60 KDM4E (0.55) HRH3HTR3EMEN1HTR3BCYP1A2
SCHEMBL2266909 0.60 CHRNB2 (0.49) HRH3HTR3EMEN1HTR3BCYP1A2
SCHEMBL1136912 0.60 AKT2 (0.47) HRH3HTR3EMEN1HTR3BCYP1A2
SCHEMBL223203 0.60 CHKA (0.59) HRH3HTR3EMEN1HTR3BCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2013211-B1 PURINE DERIVATIVES FOR USE AS ADENOSIN A2A RECEPTOR AGONISTS NOVARTIS AG (CH) 2012-03-14 EP disclosed