SCHEMBL360254

SCHEMBL360254

Oc1ccnc2ccc(Br)cc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 6/20 0.51
NCF1 P14598 1/20 0.47
ALK Q9UM73 1/20 0.45
CHEK1 O14757 1/20 0.44
PIM1 P11309 1/20 0.44
AKT1 P31749 1/20 0.44
FLT3 P36888 1/20 0.44
PIM3 Q86V86 1/20 0.44
CCNC P24863 1/20 0.44
CDK8 P49336 1/20 0.44
LMNA P02545 2/20 0.42
MAPT P10636 1/20 0.42
GAK O14976 1/20 0.42
EPHB6 O15197 1/20 0.42
RIPK2 O43353 1/20 0.42
STK16 O75716 1/20 0.42
ABL1 P00519 1/20 0.42
ACVR1 Q04771 1/20 0.42
AAK1 Q2M2I8 1/20 0.42
COQ8A Q8NI60 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1490718 0.84 ALK (0.50) SLC22A12NCF1ALKGAKHTT
SCHEMBL1332713 0.79 PARP1 (0.47) LMNAMAPTRIPK2HTTALOX15
SCHEMBL14690611 0.79 SLC22A12 (0.51) SLC22A12NCF1ALKCHEK1PIM1
SCHEMBL30819181 0.79 PARP1 (0.47) LMNAMAPTRIPK2HTTALOX15
SCHEMBL29896761 0.79 SLC22A12 (0.51) SLC22A12NCF1ALKCHEK1PIM1
SCHEMBL28140818 0.78 SMN1; SMN2 (0.44) SLC22A12NCF1ALKCHEK1PIM1
SCHEMBL3268768 0.76 NR4A2 (0.61) CCNCCDK8MAPTGAKRIPK2
SCHEMBL729828 0.76 SLC22A12 (0.49) SLC22A12NCF1ALKCHEK1PIM1
SCHEMBL5539379 0.76 HTR1A (0.54) SLC22A12FLT3PIM3CDK8LMNA
SCHEMBL591523 0.76 CDK8 (0.49) SLC22A12CCNCCDK8MAPTGAK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 192 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-120035581-A Amplifying preparation method of 6-bromo-4-hydroxyquinoline 上海再启生物技术有限公司 2025-05-23 CN claimed
US-20210246128-A1 BICYCLE TOPOISOMERASE I INHIBITING COMPOUNDS, PROCESS FOR PREPARATION AND USE THEREOF COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2021-08-12 US claimed
EP-3807248-A1 BICYCLE TOPOISOMERASE I INHIBITING COMPOUNDS, PROCESS FOR PREPARATION AND USE THEREOF Council of Scientific and Industrial Research (IN) 2021-04-21 EP claimed
US-10401747-B1 Undercoat layer for imaging device XEROX CORPORATION (US) 2019-09-03 US claimed
EP-1339690-B1 N-TYPE CALCIUM CHANNEL ANTAGONISTS FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2009-01-21 EP claimed
US-20040053965-A1 N-type calcium channel antagonists for the treatment of pain ASTRAZENECA AB (SE) 2004-03-18 US claimed
CN-121609673-B PDE4 inhibitor and preparation method and application thereof WUYI UNIVERSITY (CN) 2026-05-26 CN disclosed
WO-2026051010-A1 SCALE-UP PREPARATION METHOD FOR 6-BROMO-4-HYDROXYQUINOLINE 上海再启生物技术有限公司 2026-03-12 WO disclosed
WO-2026051010-A1 SCALE-UP PREPARATION METHOD FOR 6-BROMO-4-HYDROXYQUINOLINE 上海再启生物技术有限公司 2026-03-12 WO disclosed
US-12486234-B2 PAPD5 inhibitors and methods of use thereof CHILDREN'S MEDICAL CENTER CORPORATION (US) 2025-12-02 US disclosed
US-20250213571-A1 TYK2 INHIBITORS AND USES THEREOF ALUMIS INC. 2025-07-03 US disclosed
CN-120035581-A Amplifying preparation method of 6-bromo-4-hydroxyquinoline 上海再启生物技术有限公司 2025-05-23 CN disclosed
CN-120035581-A Amplifying preparation method of 6-bromo-4-hydroxyquinoline 上海再启生物技术有限公司 2025-05-23 CN disclosed
US-20060009460-A1 Quinoline- and isoquinoline-based compounds exhibiting ATP-utilizing enzyme inhibitory activity, and compositions, and uses thereof AGRIUS GROUP, LLC. 2006-01-12 US disclosed
WO-2005120509-A1 QUINOLINE- AND ISOQUINOLINE-BASED COMPOUNDS EXHIBITING ATP-UTILIZING ENZYME INHIBITORY ACTIVITY, AND COMPOSITIONS, AND USES THEREOF AMPHORA DISCOVERY CORPORATION (US) 2005-12-22 WO disclosed
EP-1382603-A1 NITROGENOUS FUSED−RING COMPOUND HAVING PYRAZOLYL GROUP AS SUBSTITUENT AND MEDICINAL COMPOSITION THEREOF Eisai Co., Ltd. (JP) 2004-01-21 EP disclosed
EP-0518530-B1 Improvements in or relating to excitatory amino acid receptor antagonists LILLY CO ELI (US) 1996-10-09 EP disclosed
US-5196421-A Treatment of neurological disorders ELI LILLY AND COMPANY (US) 1993-03-23 US disclosed
EP-0518530-A2 Improvements in or relating to excitatory amino acid receptor antagonists ELI LILLY AND COMPANY (US) 1992-12-16 EP disclosed
US-5153196-A Administering for reduction of neurotransmission in nervous system disorders ELI LILLY AND COMPANY (US) 1992-10-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12486234-B2 PAPD5 inhibitors and methods of use thereof POT1, PARP15, TERT SLC22A12 4275/4885NCF1 3197/4885ALK 4849/4885
US-20250213571-A1 TYK2 INHIBITORS AND USES THEREOF TYK2, JAK1, JAK2 SLC22A12 4578/4885NCF1 3570/4885ALK 914/4885
US-20060009460-A1 Quinoline- and isoquinoline-based compounds exhibiting ATP-utilizing enzyme inhibitory activity, and compositions, and uses thereof ATP5ME, ATP5MG, ATP5MK SLC22A12 2574/4885NCF1 2180/4885ALK 4689/4885
US-20040053965-A1 N-type calcium channel antagonists for the treatment of pain CACNA1B, CACNA1E, CACNA1A SLC22A12 3556/4885NCF1 334/4885ALK 4035/4885
US-20210246128-A1 BICYCLE TOPOISOMERASE I INHIBITING COMPOUNDS, PROCESS FOR PREPARATION AND USE THEREOF TOP1, TOP2A, TOP2B SLC22A12 2171/4885NCF1 1641/4885ALK 4881/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.