SCHEMBL1490718

SCHEMBL1490718

Oc1ccnc2cc(Br)ccc12

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 1/20 0.50
SLC22A12 Q96S37 6/20 0.48
CYP1A2 P05177 1/20 0.46
CYP2C19 P33261 1/20 0.46
HTT P42858 1/20 0.46
GAK O14976 1/20 0.42
PTGES O14684 1/20 0.40
PLAU P00749 2/20 0.40
ALOX15 P16050 1/20 0.40
EGFR P00533 1/20 0.39
NCF1 P14598 1/20 0.37
TLR8 Q9NR97 1/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
PLG P00747 1/20 0.37
PLAT P00750 1/20 0.37
ERN1 O75460 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9397293 0.90 SLC22A12 (0.45) ALKSLC22A12CYP1A2CYP2C19HTT
SCHEMBL360254 0.84 SLC22A12 (0.51) ALKSLC22A12CYP1A2CYP2C19HTT
SCHEMBL28164080 0.79 TLR8 (0.54) HTTALOX15EGFRTLR8KDM4E
SCHEMBL29509132 0.79 TLR8 (0.54) HTTALOX15EGFRTLR8KDM4E
SCHEMBL4470963 0.79 ALK (0.53) ALKSLC22A12CYP1A2CYP2C19HTT
SCHEMBL29896720 0.79 ALK (0.53) ALKSLC22A12CYP1A2CYP2C19HTT
SCHEMBL23498024 0.78 SLC22A12 (0.37) ALKSLC22A12CYP2C19GAKEGFR
SCHEMBL2086578 0.78 EGFR (0.53) ALKHTTGAKEGFRTLR8
Bromide SCHEMBL11522045 0.78 ALK (0.51) ALKSLC22A12CYP1A2CYP2C19HTT
SCHEMBL1496398 0.77 ALK (0.51) ALKSLC22A12CYP1A2CYP2C19HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 243 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4076459-B1 PRMT5 INHIBITORS MERCK SHARP & DOHME LLC (US) 2026-04-29 EP disclosed
US-12595248-B2 PRMT5 inhibitors MERCK SHARP & DOHME LLC (US) 2026-04-07 US disclosed
EP-4076460-B1 1,4-DIHYDRO-2H-SPIRO[ISOQUINOLINE-3,4'-PIPERIDINE DERIVATIVES AS PRMT5 INHIBITORS FOR THE TREATMENT OF CANCER MERCK SHARP & DOHME LLC (US) 2026-01-21 EP disclosed
US-12503438-B2 Compounds for the treatment of kinase-dependent disorders EXELIXIS, INC. (US) 2025-12-23 US disclosed
US-12492200-B2 NLRP3 modulators Birstol Myers-Squibb Company (US) 2025-12-09 US disclosed
WO-2025235363-A1 CYCLIN-DEPENDENT KINASE 4 DEGRADERS BLUEPRINT MEDICINES CORPORATION (US) 2025-11-13 WO disclosed
US-12441730-B2 PRMT5 inhibitors MERCK SHARP & DOHME LLC (US) 2025-10-14 US disclosed
US-20250313561-A1 NEXT-GENERATION MODULATORS OF STIMULATOR OF INTERFERON GENES (STING) RYVU THERAPEUTICS S A (PL) 2025-10-09 US disclosed
US-12391675-B2 NLRP3 modulators INNATE TUMOR IMMUNITY, INC. (US) 2025-08-19 US disclosed
US-12371428-B2 Pyridone compounds and methods of use EXELIXIS, INC. (US) 2025-07-29 US disclosed
EP-1567528-A1 MIXED LINEAGE KINASE MODULATORS ELI LILLY AND COMPANY (US) 2005-08-31 EP disclosed
WO-2005048945-A2 HYDROXYLAMINE SUBSTITUTED IMIDAZO RING COMPOUNDS 3M INNOVATIVE PROPERTIES COMPANY (US) 2005-06-02 WO disclosed
WO-2005048933-A2 OXIME SUBSTITUTED IMIDAZO RING COMPOUNDS 3M INNOVATIVE PROPERTIES COMPANY (US) 2005-06-02 WO disclosed
WO-2005018551-A2 OXIME SUBSTITUTED IMIDAZO-CONTAINING COMPOUNDS 3M INNOVATIVE PROPERTIES COMPANY (US) 2005-03-03 WO disclosed
WO-2005018556-A2 HYDROXYLAMINE SUBSTITUTED IMIDAZO-CONTAINING COMPOUNDS 3M INNOVATIVE PROPERTIES COMPANY (US) 2005-03-03 WO disclosed
US-20040147543-A1 Aryl substituted imidazoquinolines 3M INNOVATIVE PROPERTIES COMPANY 2004-07-29 US disclosed
WO-2004058759-A1 ARYL / HETARYL SUBSTITUTED IMIDAZOQUINOLINES 3M INNOVATIVE PROPERTIES COMPANY (US) 2004-07-15 WO disclosed
WO-2004048383-A1 MIXED LINEAGE KINASE MODULATORS ELI LILLY AND COMPANY (US) 2004-06-10 WO disclosed
US-4447435-A HYPOTENSIVE AGENTS THE BOOTS COMPANY PLC (GB) 1984-05-08 US disclosed
US-4442109-A 3-Methylthiomethyl-and 3-methylsulfinylmethyl-4-quinolinones useful for treating hypertension THE BOOTS COMPANY LIMITED (GB) 1984-04-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12595248-B2 PRMT5 inhibitors PRMT5, PRMT1, PRMT6 ALK 2180/4885SLC22A12 3891/4885CYP1A2 2702/4885
US-12492200-B2 NLRP3 modulators NLRP3, NLRP1, PYCARD ALK 4829/4885SLC22A12 996/4885CYP1A2 556/4885
US-12371428-B2 Pyridone compounds and methods of use PDXK, PLK2, MAP4K2 ALK 1024/4885SLC22A12 4799/4885CYP1A2 2461/4885
US-12391675-B2 NLRP3 modulators NLRP3, NLRP1, PYCARD ALK 4810/4885SLC22A12 1098/4885CYP1A2 667/4885
US-12503438-B2 Compounds for the treatment of kinase-dependent disorders ERBB2, ERBB3, PTK2B ALK 300/4885SLC22A12 3969/4885CYP1A2 4184/4885
US-20250313561-A1 NEXT-GENERATION MODULATORS OF STIMULATOR OF INTERFERON GENES (STING) STING1, IRF3, CGAS ALK 3385/4885SLC22A12 3641/4885CYP1A2 637/4885
US-12441730-B2 PRMT5 inhibitors PRMT5, PRMT1, PRMT3 ALK 1901/4885SLC22A12 2238/4885CYP1A2 1963/4885
US-20040147543-A1 Aryl substituted imidazoquinolines IL2, IFNG, IRF3 ALK 3020/4885SLC22A12 4432/4885CYP1A2 850/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.